SCHEMBL6870516

SCHEMBL6870516

COc1ccc(CNC(=O)c2cc(N)n3nc(-c4nccs4)nc3c2)cc1OC

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.46
CTSD P07339 2/20 0.44
DHFR P00374 1/20 0.44
ADORA3 P0DMS8 1/20 0.43
ADORA2A P29274 1/20 0.43
ADORA1 P30542 1/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
ALDH1A1 P00352 2/20 0.43
MEN1 O00255 1/20 0.43
GAA P10253 1/20 0.43
KMT2A Q03164 1/20 0.43
LMNA P02545 2/20 0.43
MAPK1 P28482 2/20 0.43
RECQL P46063 1/20 0.42
HSD17B10 Q99714 1/20 0.42
BCHE P06276 1/20 0.42
ACHE P22303 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6870625 0.90 MAPK10 (0.45) KDM4ESMN1; SMN2ALDH1A1GAALMNA
SCHEMBL6869924 0.90 CHRM4 (0.47) KDM4EDHFRADORA2AALDH1A1MEN1
SCHEMBL6863441 0.86 HPGD (0.45) KDM4EALDH1A1MEN1GAAKMT2A
SCHEMBL6873737 0.85 L3MBTL1 (0.43) KDM4EADORA3ADORA2AADORA1SMN1; SMN2
SCHEMBL6867467 0.85 KDM4E (0.46) KDM4EADORA2ASMN1; SMN2ALDH1A1MEN1
SCHEMBL6871432 0.81 ADORA2A (0.40) ADORA2AADORA1SMN1; SMN2ALDH1A1MEN1
SCHEMBL6867257 0.80 ADORA2A (0.55) ADORA3ADORA2AADORA1SMN1; SMN2ALDH1A1
SCHEMBL6867623 0.79 F2 (0.43) KDM4EADORA2AADORA1ALDH1A1GAA
SCHEMBL6872077 0.78 ADORA2A (0.42) KDM4EDHFRADORA2AADORA1ALDH1A1
SCHEMBL6872431 0.78 HDAC3 (0.40) KDM4EADORA2ASMN1; SMN2ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed