SCHEMBL6863613

SCHEMBL6863613

FC(F)(F)c1cccc(CN2CCN(CCNC3CCCCCC3)CC2)c1

nearest known ligand 0.62

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.62
ALDH1A1 P00352 1/20 0.62
GAA P10253 1/20 0.62
CARM1 Q86X55 3/20 0.59
PRMT6 Q96LA8 3/20 0.59
SIGMAR1 Q99720 2/20 0.53
LMNA P02545 1/20 0.51
DRD4 P21917 2/20 0.50
ACKR3 P25106 1/20 0.49
FAAH O00519 1/20 0.48
ROCK2 O75116 1/20 0.48
BCHE P06276 1/20 0.47
ACHE P22303 1/20 0.47
BACE1 P56817 1/20 0.47
CACNA1B Q00975 1/20 0.46
KCNH2 Q12809 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6864390 0.84 CXCR4 (0.47) ALDH1A1GAACARM1PRMT6ACKR3
SCHEMBL6864518 0.82 ACHE (0.57) KDM4EALDH1A1LMNADRD4ACKR3
SCHEMBL6863056 0.81 GAA (0.58) GAACARM1PRMT6SIGMAR1BCHE
SCHEMBL7109016 0.79 ACKR3 (0.49) DRD4ACKR3FAAHROCK2
SCHEMBL7187522 0.79 SIGMAR1 (0.70) KDM4EALDH1A1GAASIGMAR1DRD4
SCHEMBL4235961 0.78 ALDH1A1 (1.00) KDM4EALDH1A1GAAPRMT6SIGMAR1
SCHEMBL30341002 0.78 ALDH1A1 (1.00) KDM4EALDH1A1GAAPRMT6SIGMAR1
SCHEMBL7109288 0.77 POLB (0.63) KDM4EALDH1A1GAASIGMAR1LMNA
SCHEMBL8535362 0.77 KDM4E (0.60) KDM4EALDH1A1GAACARM1PRMT6
SCHEMBL7038365 0.77 CYP2D6 (0.49) ALDH1A1ACKR3FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5817489-A BACTERICIDES, OR CHEMICAL INTERMEDIATES THEREOF; DRUG LIBRARIES ISIS PHARMACEUTICALS, INC. (US) 1998-10-06 US claimed
US-6800444-B1 USEFUL AS ANTIBACTERIAL AND OTHER PHARMACEUTICAL AGENTS/INTERMEDIATES ISIS PHARMACEUTICALS, INC. 2004-10-05 US disclosed
US-6150129-A USEFUL AS ANTIBACTERIAL AND OTHER PHARMACEUTICAL AGENTS AND AS INTERMEDIATES FOR PREPARATION OF OTHER PHARMACEUTICAL AGENTS ISIS PHARMACEUTICALS, INC. (US) 2000-11-21 US disclosed
US-5922872-A BACTERICIDES AND DRUGS ISIS PHARMACEUTICALS, INC. (US) 1999-07-13 US disclosed
US-5817489-A BACTERICIDES, OR CHEMICAL INTERMEDIATES THEREOF; DRUG LIBRARIES ISIS PHARMACEUTICALS, INC. (US) 1998-10-06 US disclosed
US-5798360-A ANTIBACTERIAL AGENTS ISIS PHARMACEUTICALS, INC. (US) 1998-08-25 US disclosed
US-5780241-A ALTERING ELECTROCHEMICAL PROPERTIES BY DECYCLIZATION ISIS PHARMACEUTICALS, INC. (US) 1998-07-14 US disclosed
WO-1998020349-A1 COMPLEX CHEMICAL LIBRARIES ISIS PHARMACEUTICALS, INC. (US) 1998-05-14 WO disclosed
US-5731438-A BACTERICIDES; DRUGS ISIS PHARMACEUTICALS, INC. (US) 1998-03-24 US disclosed
WO-1998005332-A1 NOVEL HETEROCYCLE COMPOSITIONS ISIS PHARMACEUTICALS, INC. (US) 1998-02-12 WO disclosed