SCHEMBL7187522

SCHEMBL7187522

O=C(CN1CCN(Cc2cccc(C(F)(F)F)c2)CC1)NC1CCCCCC1

nearest known ligand 0.70

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 0.70
ACKR3 P25106 4/20 0.58
ALDH1A1 P00352 2/20 0.58
KDM4E B2RXH2 1/20 0.58
GAA P10253 1/20 0.58
DRD4 P21917 2/20 0.57
UBE2M P61081 4/20 0.55
DCUN1D1 Q96GG9 4/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6864004 0.85 ALDH1A1 (0.56) SIGMAR1ACKR3ALDH1A1
SCHEMBL6865191 0.83 CHRM2 (0.57) SIGMAR1ACKR3ALDH1A1KDM4EDRD4
SCHEMBL6865563 0.83 FAAH (0.61) SIGMAR1ALDH1A1KDM4EGAADRD4
SCHEMBL9849508 0.82 SMYD3 (0.75) SIGMAR1ACKR3ALDH1A1
SCHEMBL6865166 0.82 SIGMAR1 (0.67) SIGMAR1ALDH1A1GAA
SCHEMBL7112457 0.81 ALDH1A1 (0.57) ACKR3ALDH1A1
SCHEMBL6864686 0.80 ACKR3 (0.58) SIGMAR1ACKR3ALDH1A1KDM4E
SCHEMBL12310740 0.80 ALDH1A1 (0.63) ALDH1A1GAA
SCHEMBL6862228 0.80 SIGMAR1 (0.67) SIGMAR1ALDH1A1KDM4E
SCHEMBL6863613 0.79 KDM4E (0.62) SIGMAR1ACKR3ALDH1A1KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5817489-A BACTERICIDES, OR CHEMICAL INTERMEDIATES THEREOF; DRUG LIBRARIES ISIS PHARMACEUTICALS, INC. (US) 1998-10-06 US claimed
US-6660466-B1 Reacting reactive appendage compounds such as meta benzylic compounds or alpha-amide compounds with scaffold molecules having reactive functionalities and contacting the intermediate library with a reducing agent ISIS PHARMACEUTICALS, INC. 2003-12-09 US disclosed
US-6150129-A USEFUL AS ANTIBACTERIAL AND OTHER PHARMACEUTICAL AGENTS AND AS INTERMEDIATES FOR PREPARATION OF OTHER PHARMACEUTICAL AGENTS ISIS PHARMACEUTICALS, INC. (US) 2000-11-21 US disclosed
US-5922872-A BACTERICIDES AND DRUGS ISIS PHARMACEUTICALS, INC. (US) 1999-07-13 US disclosed
US-5817489-A BACTERICIDES, OR CHEMICAL INTERMEDIATES THEREOF; DRUG LIBRARIES ISIS PHARMACEUTICALS, INC. (US) 1998-10-06 US disclosed
US-5798360-A ANTIBACTERIAL AGENTS ISIS PHARMACEUTICALS, INC. (US) 1998-08-25 US disclosed
US-5780241-A ALTERING ELECTROCHEMICAL PROPERTIES BY DECYCLIZATION ISIS PHARMACEUTICALS, INC. (US) 1998-07-14 US disclosed
US-5731438-A BACTERICIDES; DRUGS ISIS PHARMACEUTICALS, INC. (US) 1998-03-24 US disclosed