SCHEMBL6865280

SCHEMBL6865280

Nc1ccc(-c2ccc[nH]2)c(N)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 2/20 0.38
AURKB Q96GD4 1/20 0.38
INCENP Q9NQS7 1/20 0.38
PDPK1 O15530 1/20 0.36
RET P07949 1/20 0.36
FLT3 P36888 1/20 0.36
ALK Q9UM73 1/20 0.36
CASP1 P29466 2/20 0.35
ALDH1A1 P00352 4/20 0.35
NPC1 O15118 3/20 0.35
RAB9A P51151 3/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
CYP3A4 P08684 3/20 0.35
TSHR P16473 2/20 0.35
TP53 P04637 1/20 0.35
MAPK1 P28482 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
ADORA2A P29274 1/20 0.35
LMNA P02545 3/20 0.34
PTPRC P08575 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7800798 0.84 PDPK1 (0.39) AURKAAURKBINCENPPDPK1RET
Hydrochloric Acid SCHEMBL8099675 0.82 PDPK1 (0.38) AURKAAURKBINCENPPDPK1RET
SCHEMBL5704833 0.82 TSHR (0.41) AURKAPDPK1RETFLT3ALK
SCHEMBL18755070 0.81 ALDH1A1 (0.43) AURKAPDPK1RETFLT3ALK
SCHEMBL31167504 0.81 GPR35 (0.44) AURKAAURKBINCENPPDPK1ALDH1A1
SCHEMBL28723386 0.79 ADORA2A (0.38) PDPK1RETFLT3ALKALDH1A1
SCHEMBL6137058 0.77 KDM1A (0.47) PDPK1RETFLT3ALKCASP1
SCHEMBL86365 0.77 ALDH1A1 (0.52) AURKAAURKBINCENPCASP1ALDH1A1
SCHEMBL30867600 0.77 ALDH1A1 (0.52) AURKAAURKBINCENPCASP1ALDH1A1
SCHEMBL28722142 0.77 MAOA (0.41) PDPK1RETFLT3ALKCASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6811573-B2 HAIR DYES; INTENSE, STABLE BLUE COLOR SHADES IN ADDITION TO NATURAL, PURPLE OR VIOLET ONES WELLA AKTIENGESELLSCHAFT (DE) 2004-11-02 US disclosed
US-20030093867-A1 Dyes for keratin fibres containing 1,3-diamino-4-heteroarylbenzene derivatives and novel 1,3-diamino-4-heteroarylbenzene derivatives HFC PRESTIGE INTERNATIONAL OPERATIONS SWITZERLAND SÀRL (CH) 2003-05-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030093867-A1 Dyes for keratin fibres containing 1,3-diamino-4-heteroarylbenzene derivatives and novel 1,3-diamino-4-heteroarylbenzene derivatives KRT18, DSP, TUBB4B AURKA 1360/4885AURKB 816/4885INCENP 2132/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.