SCHEMBL6869047

SCHEMBL6869047

COC(=O)c1cc(N)n2nc(-c3cccn3C)nc2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 15/20 0.40
NAMPT P43490 1/20 0.38
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
HSD17B10 Q99714 1/20 0.37
NPC1 O15118 2/20 0.37
MAPT P10636 2/20 0.37
RAB9A P51151 2/20 0.37
PKM P14618 1/20 0.36
NFKB1 P19838 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
DAPK3 O43293 1/20 0.36
JAK2 O60674 1/20 0.36
PRKD3 O94806 1/20 0.36
MAP4K4 O95819 1/20 0.36
ABL1 P00519 1/20 0.36
CSF1R P07333 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7142283 0.87 ALOX15 (0.43) ADORA2ANAMPTKDM4EALDH1A1HPGD
SCHEMBL6868263 0.82 MAPT (0.46) ADORA2ANAMPTALDH1A1NPC1MAPT
SCHEMBL6867146 0.81 ADORA2A (0.62) ADORA2AKDM4EALDH1A1HPGDMAPT
SCHEMBL6871212 0.81 ALDH1A1 (0.48) ADORA2AKDM4EALDH1A1HPGDHSD17B10
SCHEMBL6871320 0.80 SMN1; SMN2 (0.43) ADORA2ANAMPTKDM4EALDH1A1HPGD
SCHEMBL6868324 0.80 NAMPT (0.46) ADORA2ANAMPTKDM4EALDH1A1HPGD
SCHEMBL6868261 0.79 NPC1 (0.48) ADORA2AKDM4EALDH1A1HPGDHSD17B10
SCHEMBL7703259 0.78 ALDH1A1 (0.42) ADORA2ANAMPTKDM4EALDH1A1HPGD
SCHEMBL6872919 0.78 KDM4A (0.52) ADORA2AKDM4EALDH1A1HPGDHSD17B10
SCHEMBL6867096 0.77 TP53 (0.44) KDM4EALDH1A1HPGDHSD17B10MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed