SCHEMBL6868263

SCHEMBL6868263

Cn1cccc1-c1nc2cc(C(=O)Nc3ccccc3)cc(N)n2n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.46
MAPK1 P28482 1/20 0.46
TBK1 Q9UHD2 1/20 0.44
ADORA2A P29274 3/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
NAMPT P43490 1/20 0.39
POLB P06746 1/20 0.39
KDR P35968 1/20 0.38
TP53 P04637 1/20 0.38
RAB9A P51151 3/20 0.38
NPC1 O15118 2/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
JAK1 P23458 1/20 0.38
PKM P14618 1/20 0.38
NFKB1 P19838 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7142283 0.85 ALOX15 (0.43) ADORA2AMEN1KMT2ANAMPTRAB9A
SCHEMBL6868324 0.85 NAMPT (0.46) ADORA2AMEN1KMT2ANAMPTALDH1A1
SCHEMBL6868100 0.83 ADORA2A (0.44) MAPTADORA2AMEN1KMT2APOLB
SCHEMBL6869047 0.82 ADORA2A (0.40) MAPTADORA2ANAMPTKDRRAB9A
SCHEMBL6871320 0.81 SMN1; SMN2 (0.43) MAPTADORA2AMEN1KMT2ANAMPT
SCHEMBL6868261 0.80 NPC1 (0.48) MAPTADORA2APOLBTP53RAB9A
SCHEMBL6867096 0.79 TP53 (0.44) MAPTKMT2ATP53ALDH1A1LMNA
SCHEMBL6867473 0.79 KMT2A (0.43) MAPTADORA2AKMT2ANAMPTTP53
SCHEMBL6870449 0.79 RAB9A (0.45) MAPTTBK1ADORA2AMEN1KMT2A
SCHEMBL6868483 0.78 ADORA2A (0.64) ADORA2AKDRPLAU

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed