SCHEMBL6868261

SCHEMBL6868261

Cn1cccc1-c1nc2cc(C(=O)NC3CCCCC3)cc(N)n2n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.48
RAB9A P51151 3/20 0.48
KDM4E B2RXH2 3/20 0.44
HTT P42858 1/20 0.44
JAK2 O60674 1/20 0.42
JAK1 P23458 1/20 0.42
ALDH1A1 P00352 2/20 0.42
HPGD P15428 1/20 0.42
HSD17B10 Q99714 1/20 0.42
TP53 P04637 1/20 0.41
ADORA2A P29274 4/20 0.41
POLB P06746 1/20 0.41
MAPT P10636 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
LMNA P02545 1/20 0.40
TSHR P16473 1/20 0.40
CNR1 P21554 1/20 0.39
BMPR1B O00238 1/20 0.39
BMPR1A P36894 1/20 0.39
TGFBR1 P36897 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6868095 0.83 KDM4E (0.53) NPC1RAB9AKDM4EHTTALDH1A1
SCHEMBL7142283 0.80 ALOX15 (0.43) NPC1RAB9AKDM4EHTTALDH1A1
SCHEMBL6868263 0.80 MAPT (0.46) NPC1RAB9AJAK1ALDH1A1TP53
SCHEMBL6870443 0.79 LMNA (0.45) NPC1RAB9AKDM4EALDH1A1HPGD
SCHEMBL6863748 0.79 ADORA2A (0.64) NPC1RAB9AKDM4EHTTALDH1A1
SCHEMBL6871320 0.79 SMN1; SMN2 (0.43) NPC1RAB9AKDM4EHTTALDH1A1
SCHEMBL6868478 0.79 ADORA2A (0.64) NPC1RAB9AKDM4EHTTALDH1A1
SCHEMBL6869047 0.79 ADORA2A (0.40) NPC1RAB9AKDM4EJAK2ALDH1A1
SCHEMBL6867146 0.79 ADORA2A (0.62) KDM4EALDH1A1HPGDADORA2AMAPT
SCHEMBL6867550 0.78 ADORA2A (0.67) HPGDADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed