SCHEMBL6869820

SCHEMBL6869820

COc1cc(CNC(=O)c2cc(N)n3nc(-c4ccc(C)s4)nc3c2)cc(OC)c1OC

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.44
MAPK10 P53779 2/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
RAB9A P51151 1/20 0.44
HSD17B10 Q99714 2/20 0.43
PKM P14618 1/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 5/20 0.42
MAPT P10636 3/20 0.42
CHRM4 P08173 2/20 0.41
TP53 P04637 1/20 0.41
ALOX15 P16050 1/20 0.40
APOBEC3A P31941 1/20 0.40
APOBEC3G Q9HC16 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
THRB P10828 1/20 0.40
NAMPT P43490 1/20 0.40
HPGD P15428 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6872062 0.86 TP53 (0.47) KDM4EALDH1A1LMNAMAPTTP53
SCHEMBL6863351 0.85 PLAU (0.47) KDM4EHSD17B10ALDH1A1LMNAMAPT
SCHEMBL6868316 0.83 ADORA2A (0.55) KDM4EMAPK10SMN1; SMN2HSD17B10PKM
SCHEMBL6869607 0.81 ADORA2A (0.52) ALDH1A1LMNAMAPT
SCHEMBL6870625 0.81 MAPK10 (0.45) KDM4EMAPK10SMN1; SMN2RAB9AHSD17B10
SCHEMBL6869252 0.81 ADORA2A (0.57) SMN1; SMN2HSD17B10LMNAMAPTHPGD
SCHEMBL6863086 0.80 PLAU (0.44) KDM4ESMN1; SMN2HSD17B10ALDH1A1LMNA
SCHEMBL6870770 0.79 ALDH1A1 (0.41) KDM4EMAPK10SMN1; SMN2HSD17B10PKM
SCHEMBL6868343 0.78 ADORA2A (0.45) KDM4ESMN1; SMN2RAB9APKMALDH1A1
SCHEMBL6871700 0.78 SMN1; SMN2 (0.41) KDM4ESMN1; SMN2RAB9AALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed