SCHEMBL6870004

SCHEMBL6870004

COc1cccc(-c2csc(C(N)=O)c2)c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 1/20 0.64
HSD17B2 P37059 1/20 0.64
PARP1 P09874 2/20 0.51
IKBKB O14920 3/20 0.50
ALDH1A1 P00352 3/20 0.50
HSD17B10 Q99714 2/20 0.50
LMNA P02545 1/20 0.50
MAPT P10636 1/20 0.50
CDK2 P24941 1/20 0.48
IKBKE Q14164 1/20 0.48
AURKB Q96GD4 1/20 0.48
TBK1 Q9UHD2 1/20 0.48
HDAC4 P56524 1/20 0.48
HDAC8 Q9BY41 1/20 0.48
ATP4A P20648 1/20 0.47
ATP4B P51164 1/20 0.47
PLG P00747 1/20 0.46
PLAU P00749 1/20 0.46
PLAT P00750 1/20 0.46
CDC7 O00311 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6457495 0.82 ABL1 (0.52) HSD17B1HSD17B2HDAC6
SCHEMBL30916784 0.78 TUBB4A (0.58) HSD17B1HSD17B2MAPTHTT
SCHEMBL26044573 0.78 NPC1 (0.55) HSD17B1HSD17B2ALDH1A1HSD17B10LMNA
SCHEMBL5605556 0.77 HDAC6 (0.62) IKBKBPLAUHDAC6
SCHEMBL5613367 0.77 HDAC6 (0.71) HSD17B1HSD17B2PARP1IKBKBHDAC6
SCHEMBL1690557 0.76 PARP1 (0.80) HSD17B2PARP1IKBKBHDAC4HDAC8
SCHEMBL1981372 0.76 ALDH1A1 (0.52) HSD17B1HSD17B2ALDH1A1HSD17B10LMNA
SCHEMBL25399545 0.76 KMT2A (0.54) PARP1IKBKBMAPTCDK2IKBKE
SCHEMBL4995249 0.75 PLAU (0.67) HSD17B2PARP1HDAC4HDAC8PLG
SCHEMBL30958376 0.75 PLAU (0.67) HSD17B2PARP1HDAC4HDAC8PLG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1394159-A1 New thiophene derivatives, process for their preparation and pharmaceutical compositions containing them Warner-Lambert Company LLC (US) 2004-03-03 EP claimed