SCHEMBL6870820

SCHEMBL6870820

CCOC(=O)CCN(C1(C(=O)NO)CCOCC1)S(=O)(=O)c1ccc(Oc2ccccc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 19/20 0.58
MMP13 P45452 16/20 0.52
MMP2 P08253 7/20 0.52
MMP9 P14780 6/20 0.52
MMP3 P08254 5/20 0.52
MMP8 P22894 5/20 0.52
MMP14 P50281 7/20 0.48
MMP7 P09237 2/20 0.43
ADAM17 P78536 2/20 0.43
ABCB11 O95342 1/20 0.43
MMP10 P09238 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3921083 0.93 MMP1 (0.55) MMP1MMP13MMP2MMP9MMP3
SCHEMBL6813262 0.92 MMP1 (0.67) MMP1MMP13MMP2MMP9MMP3
SCHEMBL6813516 0.92 MMP1 (0.54) MMP1MMP13MMP2MMP9MMP3
SCHEMBL6693057 0.92 MMP1 (0.68) MMP1MMP13MMP2MMP9MMP3
SCHEMBL6873149 0.90 MMP1 (0.70) MMP1MMP13MMP2MMP9MMP3
SCHEMBL7347709 0.85 MMP1 (0.56) MMP1MMP13MMP2MMP9MMP3
SCHEMBL7352211 0.85 MMP1 (0.45) MMP1MMP13MMP2MMP9MMP3
SCHEMBL3914707 0.84 MMP1 (0.63) MMP1MMP13MMP2MMP9MMP3
SCHEMBL13898990 0.84 MMP1 (0.58) MMP1MMP13MMP2MMP9MMP3
SCHEMBL3987272 0.84 MMP1 (0.68) MMP1MMP13MMP2MMP9MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1088550-A1 alpha-sulfonylamino hydroxamic acid inhibitors of matrix metallo-proteinases for the treatment of peripheral or central nervous system disorders Pfizer Products Inc. (US) 2001-04-04 EP claimed
EP-1415984-A1 Aryloxyarylsulfonylamino hydroxamic acid derivatives Pfizer Products Inc. (US) 2004-05-06 EP disclosed
US-6417229-B1 ENZYME INHIBITORS PFIZER INC 2002-07-09 US disclosed
EP-1088550-A1 alpha-sulfonylamino hydroxamic acid inhibitors of matrix metallo-proteinases for the treatment of peripheral or central nervous system disorders Pfizer Products Inc. (US) 2001-04-04 EP disclosed
EP-1003720-A1 ARYLOXYARYLSULFONYLAMINO HYDROXAMIC ACID DERIVATIVES Pfizer Products Inc. (US) 2000-05-31 EP disclosed
WO-1999007675-A1 ARYLOXYARYLSULFONYLAMINO HYDROXAMIC ACID DERIVATIVES PFIZER PRODUCTS INC. (US) 1999-02-18 WO disclosed