SCHEMBL6871806

SCHEMBL6871806

COC(=O)c1cc(N)n2nc(-c3ccoc3)nc2c1

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 17/20 0.42
ADORA3 P0DMS8 2/20 0.39
ADORA2B P29275 2/20 0.39
ADORA1 P30542 2/20 0.38
NR4A2 P43354 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6863099 0.85 ADORA2A (0.45) ADORA2AADORA3ADORA1
SCHEMBL6871212 0.83 ALDH1A1 (0.48) ADORA2A
SCHEMBL6867154 0.81 ADORA2A (0.63) ADORA2AADORA3ADORA2BADORA1
SCHEMBL6869842 0.80 PLAU (0.48) ADORA2A
SCHEMBL6870530 0.80 ADORA2A (0.43) ADORA2AADORA3ADORA2BADORA1
SCHEMBL6869244 0.80 ADORA2A (0.67) ADORA2A
SCHEMBL6867888 0.79 ADORA2A (0.66) ADORA2AADORA3ADORA2BADORA1
SCHEMBL6870631 0.79 LMNA (0.48) ADORA2AADORA3ADORA2BADORA1
SCHEMBL6871623 0.79 ADORA2A (0.67) ADORA2A
SCHEMBL6863797 0.78 ADORA2A (0.50) ADORA2AADORA3ADORA2BADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed