SCHEMBL6870530

SCHEMBL6870530

CCCCNC(=O)c1cc(N)n2nc(-c3ccoc3)nc2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 9/20 0.43
EGLN2 Q96KS0 1/20 0.41
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
POLB P06746 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
ALOX15 P16050 1/20 0.40
CASP1 P29466 1/20 0.40
BLM P54132 1/20 0.40
CASP7 P55210 1/20 0.40
KMT2A Q03164 1/20 0.40
MCL1 Q07820 1/20 0.40
HSD17B10 Q99714 1/20 0.40
CTDSP1 Q9GZU7 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
FYN P06241 1/20 0.39
ADORA1 P30542 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6866973 0.85 BACE1 (0.48) EGLN2KDM4EALDH1A1POLBMAPT
SCHEMBL6870605 0.82 ADORA2A (0.58) ADORA2AKDM4EMEN1ALDH1A1POLB
SCHEMBL6869746 0.82 PLAU (0.43) ADORA2AKDM4EMEN1ALDH1A1POLB
SCHEMBL6867215 0.81 PLAU (0.47) MEN1POLBHPGDKMT2ASMN1; SMN2
SCHEMBL6871283 0.80 PTGER2 (0.44) ADORA2AMEN1ALDH1A1POLBMAPT
SCHEMBL6872215 0.80 EGLN2 (0.42) ADORA2AEGLN2KDM4EALDH1A1MAPT
SCHEMBL6870649 0.80 ADORA2A (0.61) ADORA2ASMN1; SMN2
SCHEMBL6871806 0.80 ADORA2A (0.42) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL6869803 0.80 ADORA2A (0.41) ADORA2AMEN1POLBKMT2AKDR
SCHEMBL6863099 0.79 ADORA2A (0.45) ADORA2AADORA1ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed