SCHEMBL6872018

SCHEMBL6872018

COc1ccc(-c2nc3cc(C(=O)NC4CC4)cc(N)n3n2)s1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 8/20 0.41
CHRM4 P08173 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
ALDH1A1 P00352 1/20 0.36
SMYD3 Q9H7B4 2/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
KDM4E B2RXH2 1/20 0.36
MAPT P10636 1/20 0.36
MAPK11 Q15759 1/20 0.36
MAPK14 Q16539 1/20 0.36
LMNA P02545 1/20 0.36
HPGDS O60760 2/20 0.36
TP53 P04637 1/20 0.36
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6869677 0.96 ADORA2A (0.42) ADORA2AMEN1KMT2ALMNAHPGDS
SCHEMBL6873063 0.95 MEN1 (0.44) ADORA2AMEN1KMT2AALDH1A1RAB9A
SCHEMBL6869619 0.95 MEN1 (0.44) ADORA2AMEN1KMT2AALDH1A1RAB9A
SCHEMBL6871503 0.84 ADORA2A (0.43) ADORA2AALDH1A1NPC1RAB9AKDM4E
SCHEMBL6873034 0.84 ADORA2A (0.39) ADORA2AALDH1A1NPC1RAB9AKDM4E
SCHEMBL6869680 0.83 ADORA2A (0.39) ADORA2AALDH1A1NPC1RAB9AKDM4E
SCHEMBL6870443 0.83 LMNA (0.45) ADORA2AMEN1KMT2AALDH1A1NPC1
SCHEMBL6867527 0.83 ADORA2A (0.38) ADORA2AKMT2AALDH1A1NPC1RAB9A
SCHEMBL6869624 0.82 ADORA2A (0.41) ADORA2AMEN1KMT2AALDH1A1NPC1
SCHEMBL6863144 0.81 NAAA (0.39) ADORA2AMEN1KMT2ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed