SCHEMBL6874191

SCHEMBL6874191

COc1ccc2[nH]cc(CNC3CCC(Nc4nc5c(c(N(C)C)n4)CCCC5)CC3)c2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 5/20 0.44
ACHE P22303 3/20 0.44
HTR1A P08908 3/20 0.40
HTR1B P28222 3/20 0.40
HTR4 Q13639 2/20 0.40
HTR2A P28223 2/20 0.40
HTR3E A5X5Y0 1/20 0.40
HTR3B O95264 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
HTR1D P28221 1/20 0.40
HTR2C P28335 1/20 0.40
HTR1E P28566 1/20 0.40
HTR1F P30939 1/20 0.40
HTR7 P34969 1/20 0.40
HTR2B P41595 1/20 0.40
HTR3A P46098 1/20 0.40
HTR5A P47898 1/20 0.40
MTNR1A P48039 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6458578 1.00 BCHE (0.44) BCHEACHEHTR1AHTR1BHTR4
SCHEMBL6878474 0.90 BCHE (0.43) BCHEACHEHTR1AHTR1BHTR4
SCHEMBL6456848 0.90 BCHE (0.43) BCHEACHEHTR1AHTR1BHTR4
SCHEMBL6457965 0.88 ADRA2A (0.46) BCHEACHEHTR1AHTR2AMTNR1A
SCHEMBL6874250 0.88 ADRA2A (0.46) BCHEACHEHTR1AHTR2AMTNR1A
SCHEMBL6467595 0.86 LMNA (0.53) BCHEACHEHTR1ALMNAALDH1A1
SCHEMBL6875174 0.86 LMNA (0.53) BCHEACHEHTR1ALMNAALDH1A1
SCHEMBL6459434 0.84 MCHR1 (0.41) BCHEACHEL3MBTL1LMNAKDM4E
SCHEMBL6875761 0.84 MCHR1 (0.41) BCHEACHEL3MBTL1LMNAKDM4E
SCHEMBL6874201 0.84 ADRA2A (0.45) CYP1A2CYP2D6L3MBTL1LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed