SCHEMBL6874339

SCHEMBL6874339

CN(C)c1nc(NC2CCC(NC(=O)OCc3ccc([N+](=O)[O-])cc3)CC2)nc2c1CCCC2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 4/20 0.44
MCHR1 Q99705 4/20 0.44
EPHX1 P07099 3/20 0.44
MEN1 O00255 1/20 0.38
MAPT P10636 1/20 0.38
HTT P42858 1/20 0.38
KMT2A Q03164 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
HRH1 P35367 3/20 0.37
HTR2B P41595 3/20 0.37
ALDH1A1 P00352 3/20 0.37
GAA P10253 1/20 0.37
ACHE P22303 1/20 0.37
CACNB4 O00305 1/20 0.37
CACNA1A O00555 1/20 0.37
CACNA1G O43497 1/20 0.37
CACNG3 O60359 1/20 0.37
CACNA1F O60840 1/20 0.37
CACNA1H O95180 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6876882 0.90 MCHR1 (0.39) ADRA2AMCHR1EPHX1MEN1MAPT
SCHEMBL7046594 0.88 ALDH1A1 (0.50) ADRA2AMCHR1EPHX1MEN1KMT2A
SCHEMBL6868112 0.85 MCHR1 (0.56) ADRA2AMCHR1MAPTHTTKMT2A
SCHEMBL6868116 0.85 MCHR1 (0.56) ADRA2AMCHR1MAPTHTTKMT2A
SCHEMBL4030186 0.84 MCHR1 (0.64) ADRA2AMCHR1HRH1HTR2BALDH1A1
SCHEMBL4030189 0.84 MCHR1 (0.64) ADRA2AMCHR1HRH1HTR2BALDH1A1
SCHEMBL6458129 0.84 ADRA2A (0.44) ADRA2AMCHR1EPHX1MAPTHRH1
SCHEMBL6458136 0.84 ADRA2A (0.44) ADRA2AMCHR1EPHX1MAPTHRH1
SCHEMBL6877509 0.84 MCHR1 (0.40) ADRA2AMCHR1HTTSMN1; SMN2HRH1
SCHEMBL6868077 0.82 MCHR1 (0.43) ADRA2AMCHR1EPHX1MEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed