SCHEMBL6875745

SCHEMBL6875745

CN(Cc1ccc(F)cc1F)C(=O)c1nc(-c2c(F)cccc2F)[nH]c(=O)c1O

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 2/20 0.42
ATM Q13315 1/20 0.36
ERCC1 P07992 4/20 0.36
FEN1 P39748 4/20 0.36
ERCC4 Q92889 4/20 0.36
RNASEH1 O60930 1/20 0.36
PIN1 Q13526 2/20 0.35
CYP1A1 P04798 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP1B1 Q16678 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6882031 0.90 SLC6A4 (0.36) RIPK1ATMERCC1FEN1ERCC4
SCHEMBL6883583 0.87 ERCC1 (0.44) ATMERCC1FEN1ERCC4PIN1
SCHEMBL6886242 0.85 HSP90AA1 (0.40) ATMERCC1FEN1ERCC4RNASEH1
SCHEMBL6882008 0.83 ERCC1 (0.37) RIPK1ATMERCC1FEN1ERCC4
SCHEMBL6884260 0.83 PIN1 (0.41) ERCC1FEN1ERCC4RNASEH1PIN1
SCHEMBL6885172 0.82 PIN1 (0.43) ERCC1FEN1ERCC4PIN1
SCHEMBL6881498 0.81 PIN1 (0.39) ERCC1FEN1ERCC4RNASEH1PIN1
SCHEMBL6886352 0.81 PIN1 (0.46) ERCC1FEN1ERCC4PIN1
SCHEMBL6883448 0.80 RNASEH1 (0.44) ERCC1FEN1ERCC4RNASEH1PIN1
SCHEMBL6882913 0.80 TACR1 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004096128-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-11 WO disclosed