SCHEMBL6883448

SCHEMBL6883448

CN(Cc1ccc(Cl)c(Cl)c1)C(=O)c1nc(-c2c(F)cccc2F)[nH]c(=O)c1O

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
RNASEH1 O60930 1/20 0.44
PIN1 Q13526 2/20 0.41
CENPE Q02224 5/20 0.40
TRPV1 Q8NER1 1/20 0.40
ALDH1A1 P00352 1/20 0.37
ERCC1 P07992 1/20 0.37
FEN1 P39748 1/20 0.37
ERCC4 Q92889 1/20 0.37
APOBEC3A P31941 1/20 0.37
APOBEC3G Q9HC16 1/20 0.37
PSEN1 P49768 1/20 0.37
PSEN2 P49810 1/20 0.37
APH1B Q8WW43 1/20 0.37
NCSTN Q92542 1/20 0.37
APH1A Q96BI3 1/20 0.37
PSENEN Q9NZ42 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6883616 0.93 PIN1 (0.40) RNASEH1PIN1ALDH1A1ERCC1FEN1
SCHEMBL6884260 0.89 PIN1 (0.41) RNASEH1PIN1ERCC1FEN1ERCC4
SCHEMBL6886352 0.89 PIN1 (0.46) PIN1ALDH1A1ERCC1FEN1ERCC4
SCHEMBL6881498 0.87 PIN1 (0.39) RNASEH1PIN1ERCC1FEN1ERCC4
SCHEMBL6883583 0.87 ERCC1 (0.44) PIN1ERCC1FEN1ERCC4
SCHEMBL6017817 0.87 RNASEH1 (0.43) RNASEH1PIN1CENPETRPV1
SCHEMBL6885172 0.86 PIN1 (0.43) PIN1ERCC1FEN1ERCC4
SCHEMBL6885510 0.85 PIN1 (0.54) RNASEH1PIN1ERCC1FEN1ERCC4
SCHEMBL6884192 0.85 PIN1 (0.37) PIN1ERCC1FEN1ERCC4
SCHEMBL6885455 0.83 MEN1 (0.42) PIN1ERCC1FEN1ERCC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004096128-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-11 WO claimed
WO-2004096128-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-11 WO disclosed