SCHEMBL6883583

SCHEMBL6883583

CN(Cc1ccc(F)cc1)C(=O)c1nc(-c2c(F)cccc2F)[nH]c(=O)c1O

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ERCC1 P07992 3/20 0.44
FEN1 P39748 3/20 0.44
ERCC4 Q92889 3/20 0.44
PIN1 Q13526 2/20 0.43
TDP1 Q9NUW8 1/20 0.40
ATM Q13315 1/20 0.40
NSD2 O96028 1/20 0.39
KMT2A Q03164 1/20 0.39
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6885172 0.93 PIN1 (0.43) ERCC1FEN1ERCC4PIN1
SCHEMBL6886352 0.92 PIN1 (0.46) ERCC1FEN1ERCC4PIN1
SCHEMBL6885455 0.90 MEN1 (0.42) ERCC1FEN1ERCC4PIN1KMT2A
SCHEMBL6884260 0.90 PIN1 (0.41) ERCC1FEN1ERCC4PIN1KMT2A
SCHEMBL6883598 0.89 TNKS (0.43) ERCC1FEN1ERCC4PIN1ATM
SCHEMBL6881498 0.88 PIN1 (0.39) ERCC1FEN1ERCC4PIN1
SCHEMBL6883448 0.87 RNASEH1 (0.44) ERCC1FEN1ERCC4PIN1
SCHEMBL6875745 0.87 RIPK1 (0.42) ERCC1FEN1ERCC4PIN1ATM
SCHEMBL6885410 0.86 PIN1 (0.60) ERCC1FEN1ERCC4PIN1TDP1
SCHEMBL6884192 0.85 PIN1 (0.37) ERCC1FEN1ERCC4PIN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004096128-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-11 WO claimed
WO-2004096128-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-11 WO disclosed