SCHEMBL6876322

SCHEMBL6876322

COc1ccc(CNC2CCC(Nc3nc4c(c(N(C)C)n3)CCCC4)CC2)c(OC)c1OC

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 3/20 0.42
MCHR1 Q99705 3/20 0.42
APP P05067 3/20 0.39
BCHE P06276 2/20 0.35
ACHE P22303 2/20 0.35
BACE1 P56817 1/20 0.35
KDM4E B2RXH2 4/20 0.34
MEN1 O00255 1/20 0.34
GAA P10253 1/20 0.34
HTT P42858 1/20 0.34
KMT2A Q03164 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
MAPT P10636 3/20 0.34
LMNA P02545 2/20 0.34
POLB P06746 2/20 0.34
TP53 P04637 2/20 0.34
ALDH1A1 P00352 3/20 0.33
TUBB3 Q13509 1/20 0.33
NPY5R Q15761 1/20 0.33
EHMT2 Q96KQ7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6876315 1.00 ADRA2A (0.42) ADRA2AMCHR1APPBCHEACHE
SCHEMBL6867923 0.89 MCHR1 (0.45) ADRA2AMCHR1APPBCHEACHE
SCHEMBL6867919 0.89 MCHR1 (0.45) ADRA2AMCHR1APPBCHEACHE
SCHEMBL6877262 0.87 ADRA2A (0.48) ADRA2AMCHR1APPBCHEACHE
SCHEMBL6460350 0.87 ADRA2A (0.48) ADRA2AMCHR1APPBCHEACHE
SCHEMBL6874187 0.86 ADRA2A (0.45) ADRA2AMCHR1KDM4EMEN1GAA
SCHEMBL6875761 0.86 MCHR1 (0.41) ADRA2AMCHR1APPBCHEACHE
SCHEMBL6874201 0.86 ADRA2A (0.45) ADRA2AMCHR1KDM4EMEN1GAA
SCHEMBL6459434 0.86 MCHR1 (0.41) ADRA2AMCHR1APPBCHEACHE
SCHEMBL6875692 0.85 ALDH1A1 (0.52) ADRA2AMCHR1APPBCHEACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed