SCHEMBL6878302

SCHEMBL6878302

CN(Cc1ccc(Cl)c(Cl)c1)C(=O)c1nc(-c2ccc(F)cc2S(C)(=O)=O)[nH]c(=O)c1O

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RNASEH1 O60930 1/20 0.40
CENPE Q02224 5/20 0.38
ADORA2B P29275 1/20 0.37
ADORA1 P30542 1/20 0.37
ERCC1 P07992 1/20 0.35
FEN1 P39748 1/20 0.35
ERCC4 Q92889 1/20 0.35
ROCK2 O75116 1/20 0.35
PTGES O14684 1/20 0.34
WDR5 P61964 1/20 0.34
PIN1 Q13526 1/20 0.34
GSK3B P49841 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6883233 0.91 ATM (0.39) ERCC1FEN1ERCC4PIN1
SCHEMBL6886326 0.89 ERCC1 (0.36) ERCC1FEN1ERCC4PIN1
SCHEMBL6883811 0.83 RNASEH1 (0.41) RNASEH1ADORA2BADORA1PIN1
SCHEMBL6883448 0.79 RNASEH1 (0.44) RNASEH1CENPEERCC1FEN1ERCC4
SCHEMBL6884173 0.79 HTR1A (0.43) RNASEH1ERCC1FEN1ERCC4PIN1
SCHEMBL6883024 0.79 RNASEH1 (0.44) RNASEH1ERCC1FEN1ERCC4ROCK2
SCHEMBL6885510 0.78 PIN1 (0.54) RNASEH1ERCC1FEN1ERCC4PIN1
SCHEMBL6884051 0.77 RNASEH1 (0.46) RNASEH1CENPEERCC1FEN1ERCC4
SCHEMBL6885308 0.76 PIN1 (0.38) RNASEH1PIN1
SCHEMBL6017817 0.76 RNASEH1 (0.43) RNASEH1CENPEPIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004096128-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-11 WO claimed
WO-2004096128-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-11 WO disclosed