SCHEMBL6885308

SCHEMBL6885308

Cc1ccc(CN(C)C(=O)c2nc(-c3ccccc3S(=O)(=O)N(C)C)[nH]c(=O)c2O)cc1Cl

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 2/20 0.38
RNASEH1 O60930 1/20 0.36
ALDH1A1 P00352 3/20 0.35
LMNA P02545 2/20 0.35
MAPT P10636 1/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
KCNJ6 P48051 2/20 0.35
KCNJ5 P48544 2/20 0.35
KCNJ3 P48549 2/20 0.35
HSP90AA1 P07900 3/20 0.34
SLC9A1 P19634 1/20 0.34
TSPO P30536 1/20 0.34
POLB P06746 1/20 0.34
THRB P10828 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6883811 0.93 RNASEH1 (0.41) PIN1RNASEH1ALDH1A1LMNAMAPT
SCHEMBL6878297 0.92 PIN1 (0.38) PIN1RNASEH1
SCHEMBL6883865 0.86 PIN1 (0.40) PIN1RNASEH1TSPO
SCHEMBL6884448 0.85 PIN1 (0.41) PIN1ALDH1A1LMNAMAPT
SCHEMBL6883984 0.84 HTR7 (0.41) PIN1RNASEH1HSP90AA1SLC9A1
SCHEMBL6877025 0.84 PIN1 (0.53) PIN1RNASEH1
SCHEMBL6878396 0.81 PTGES (0.41) PIN1LMNA
SCHEMBL6883326 0.81 ALDH1A1 (0.44) PIN1RNASEH1ALDH1A1LMNAMAPT
SCHEMBL6883616 0.80 PIN1 (0.40) PIN1RNASEH1ALDH1A1HSP90AA1
SCHEMBL6882673 0.79 ERCC1 (0.42) PIN1RNASEH1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004096128-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-11 WO claimed
WO-2004096128-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-11 WO disclosed