SCHEMBL6880103

SCHEMBL6880103

CSc1ccc(NC(=O)N[C@H]2CC[C@@H](Nc3cc(N(C)C)c4ccccc4n3)CC2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.48
MAPT P10636 2/20 0.43
RXFP1 Q9HBX9 1/20 0.43
HTR2B P41595 2/20 0.43
HTR2C P28335 1/20 0.43
MCHR1 Q99705 4/20 0.42
EPHX1 P07099 2/20 0.41
NOX1 Q9Y5S8 1/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
KDR P35968 1/20 0.40
ADRA2A P08913 3/20 0.40
S1PR1 P21453 1/20 0.40
OPRD1 P41143 1/20 0.40
KDM4E B2RXH2 1/20 0.40
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HTR1A P08908 1/20 0.40
ADRA1A P35348 1/20 0.40
HRH1 P35367 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6880110 1.00 SIGMAR1 (0.48) SIGMAR1MAPTRXFP1HTR2BHTR2C
SCHEMBL6878072 0.89 NPC1 (0.44) SIGMAR1MAPTHTR2BHTR2CMCHR1
SCHEMBL6878067 0.89 NPC1 (0.44) SIGMAR1MAPTHTR2BHTR2CMCHR1
SCHEMBL6877589 0.87 EPHX1 (0.53) MAPTMCHR1EPHX1KDRADRA2A
SCHEMBL6878657 0.86 EPHX1 (0.49) MCHR1EPHX1ADRA2AS1PR1OPRD1
SCHEMBL6878665 0.86 EPHX1 (0.49) MCHR1EPHX1ADRA2AS1PR1OPRD1
SCHEMBL6880550 0.84 MAPT (0.54) MAPTMCHR1NPC1KDRADRA2A
SCHEMBL6880545 0.84 MAPT (0.54) MAPTMCHR1NPC1KDRADRA2A
SCHEMBL6874686 0.83 RAB9A (0.53) MAPTRXFP1NPC1RAB9AKDM4E
SCHEMBL6873468 0.83 SMN1; SMN2 (0.51) MAPTNPC1RAB9AKDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed