SCHEMBL6880113

SCHEMBL6880113

CN(C)c1ccnc(NC2CCC(NC(=O)CCc3ccccc3O)CC2)n1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.42
MTNR1B P49286 1/20 0.42
HPGD P15428 1/20 0.42
HTT P42858 1/20 0.42
RECQL P46063 1/20 0.42
MCHR1 Q99705 8/20 0.40
CNR2 P34972 7/20 0.40
CNR1 P21554 5/20 0.40
CYP2C9 P11712 1/20 0.39
CCNE1 P24864 1/20 0.39
CDK2 P24941 1/20 0.39
MAPK8 P45983 1/20 0.39
MAPK9 P45984 1/20 0.39
MAPK10 P53779 1/20 0.39
ADRA2A P08913 2/20 0.39
HRH1 P35367 2/20 0.39
HTR2B P41595 2/20 0.39
ADRA1A P35348 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6880107 1.00 MTNR1A (0.42) MTNR1AMTNR1BHPGDHTTRECQL
SCHEMBL6877817 0.90 MCHR1 (0.43) HPGDMCHR1CNR2CNR1MAPK8
SCHEMBL6877812 0.90 MCHR1 (0.43) HPGDMCHR1CNR2CNR1MAPK8
SCHEMBL6877124 0.87 EPHX2 (0.47) MCHR1CYP2C9CCNE1CDK2MAPK8
SCHEMBL6877131 0.87 EPHX2 (0.47) MCHR1CYP2C9CCNE1CDK2MAPK8
SCHEMBL6868909 0.82 SIGMAR1 (0.46) MCHR1CYP2C9CCNE1CDK2MAPK8
SCHEMBL6868904 0.82 SIGMAR1 (0.46) MCHR1CYP2C9CCNE1CDK2MAPK8
SCHEMBL6874860 0.82 ALDH1A1 (0.41) MCHR1CYP2C9CCNE1CDK2MAPK8
SCHEMBL6874855 0.82 ALDH1A1 (0.41) MCHR1CYP2C9CCNE1CDK2MAPK8
SCHEMBL6874044 0.81 AURKA (0.50) MCHR1CYP2C9CCNE1CDK2MAPK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed