SCHEMBL6880509

SCHEMBL6880509

[NH]c1ccc(CCn2cnnn2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.52
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
HRH3 Q9Y5N1 1/20 0.50
HMOX1 P09601 1/20 0.42
MAPK1 P28482 2/20 0.39
KDM4E B2RXH2 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
TP53 P04637 3/20 0.38
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37
RAB9A P51151 1/20 0.36
LTA4H P09960 1/20 0.36
KCNJ1 P48048 1/20 0.35
KCNH2 Q12809 1/20 0.35
MAPT P10636 1/20 0.34
POLB P06746 1/20 0.33
LMNA P02545 1/20 0.33
THRB P10828 1/20 0.33
HTR1A P08908 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29788842 0.82 RAB9A (0.52) ALDH1A1MEN1KMT2AHRH3HMOX1
SCHEMBL8727211 0.73 HRH3 (0.43) ALDH1A1MEN1KMT2AHRH3HMOX1
SCHEMBL29788848 0.71 HMOX1 (0.56) ALDH1A1MEN1KMT2AHMOX1TP53
SCHEMBL29788855 0.71 MEN1 (0.57) ALDH1A1MEN1KMT2AKDM4ECYP1A2
SCHEMBL9872854 0.70 MAOA (0.47) ALDH1A1MEN1KMT2AHRH3HMOX1
SCHEMBL3643462 0.65
SCHEMBL29061272 0.65
SCHEMBL10066409 0.64 MEN1 (0.54) ALDH1A1MEN1KMT2AHRH3HMOX1
SCHEMBL28609350 0.63
SCHEMBL28611936 0.63

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832091-B1 C-4' MODIFIED ADENOSINE KINASE INHIBITORS GENSIA SICOR INC (US) 2004-01-14 EP disclosed