SCHEMBL6884192

SCHEMBL6884192

CN(Cc1ccc(C(F)(F)F)c(F)c1)C(=O)c1nc(-c2c(F)cccc2F)[nH]c(=O)c1O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 2/20 0.37
HDAC3 O15379 3/20 0.37
HDAC4 P56524 3/20 0.37
HDAC6 Q9UBN7 3/20 0.37
HDAC1 Q13547 2/20 0.37
TUBB4A P04350 1/20 0.37
TUBB P07437 1/20 0.37
TUBA3C P0DPH7 1/20 0.37
TUBA1B P68363 1/20 0.37
TUBA4A P68366 1/20 0.37
TUBB4B P68371 1/20 0.37
TUBB3 Q13509 1/20 0.37
TUBB2A Q13885 1/20 0.37
TUBB8 Q3ZCM7 1/20 0.37
TUBA3E Q6PEY2 1/20 0.37
TUBA1A Q71U36 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC10 Q969S8 1/20 0.37
HDAC11 Q96DB2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6884260 0.89 PIN1 (0.41) PIN1ERCC1FEN1ERCC4MEN1
SCHEMBL6885455 0.88 MEN1 (0.42) PIN1ERCC1FEN1ERCC4MEN1
SCHEMBL6882913 0.87 TACR1 (0.46)
SCHEMBL6881498 0.86 PIN1 (0.39) PIN1ERCC1FEN1ERCC4
SCHEMBL6883583 0.85 ERCC1 (0.44) PIN1ERCC1FEN1ERCC4KMT2A
SCHEMBL6883448 0.85 RNASEH1 (0.44) PIN1ERCC1FEN1ERCC4
SCHEMBL6885172 0.84 PIN1 (0.43) PIN1ERCC1FEN1ERCC4
SCHEMBL6882031 0.84 SLC6A4 (0.36) ERCC1FEN1ERCC4KMT2A
SCHEMBL6886352 0.84 PIN1 (0.46) PIN1ERCC1FEN1ERCC4
SCHEMBL6883616 0.83 PIN1 (0.40) PIN1ERCC1FEN1ERCC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004096128-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-11 WO claimed
WO-2004096128-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-11 WO disclosed