SCHEMBL6885455

SCHEMBL6885455

CN(Cc1ccc(C(F)(F)F)cc1)C(=O)c1nc(-c2c(F)cccc2F)[nH]c(=O)c1O

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
PIN1 Q13526 2/20 0.41
TNKS O95271 3/20 0.39
TNKS2 Q9H2K2 3/20 0.39
PARP1 P09874 2/20 0.39
ERCC1 P07992 2/20 0.39
FEN1 P39748 2/20 0.39
ERCC4 Q92889 2/20 0.39
MTOR P42345 1/20 0.38
SIRT2 Q8IXJ6 1/20 0.38
PARP2 Q9UGN5 1/20 0.37
PPARA Q07869 1/20 0.37
TACR1 P25103 1/20 0.37
MLYCD O95822 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6882913 0.91 TACR1 (0.46) TACR1
SCHEMBL6883583 0.90 ERCC1 (0.44) KMT2APIN1ERCC1FEN1ERCC4
SCHEMBL6885172 0.89 PIN1 (0.43) PIN1ERCC1FEN1ERCC4
SCHEMBL6886352 0.88 PIN1 (0.46) PIN1ERCC1FEN1ERCC4
SCHEMBL6884192 0.88 PIN1 (0.37) MEN1KMT2APIN1ERCC1FEN1
SCHEMBL6884260 0.86 PIN1 (0.41) MEN1KMT2APIN1ERCC1FEN1
SCHEMBL6881498 0.84 PIN1 (0.39) PIN1ERCC1FEN1ERCC4
SCHEMBL6883448 0.83 RNASEH1 (0.44) PIN1ERCC1FEN1ERCC4
SCHEMBL6883616 0.82 PIN1 (0.40) PIN1ERCC1FEN1ERCC4
SCHEMBL6882031 0.81 SLC6A4 (0.36) KMT2AERCC1FEN1ERCC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004096128-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-11 WO claimed
WO-2004096128-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-11 WO disclosed