SCHEMBL6884448

SCHEMBL6884448

CN(Cc1ccc(F)cc1)C(=O)c1nc(-c2ccccc2S(=O)(=O)N(C)C)[nH]c(=O)c1O

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 2/20 0.41
ERCC1 P07992 2/20 0.40
FEN1 P39748 2/20 0.40
ERCC4 Q92889 2/20 0.40
ATM Q13315 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
USP1 O94782 1/20 0.38
KMT2A Q03164 1/20 0.37
LIMK2 P53671 1/20 0.37
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6878297 0.87 PIN1 (0.38) PIN1ERCC1FEN1ERCC4KMT2A
SCHEMBL6883811 0.86 RNASEH1 (0.41) PIN1ALDH1A1LMNAMAPT
SCHEMBL6885308 0.85 PIN1 (0.38) PIN1ALDH1A1LMNAMAPT
SCHEMBL6885442 0.85 PIN1 (0.43) PIN1ERCC1FEN1ERCC4ATM
SCHEMBL6883233 0.84 ATM (0.39) PIN1ERCC1FEN1ERCC4ATM
SCHEMBL6884321 0.84 HSD17B1 (0.44) PIN1ERCC1FEN1ERCC4ATM
SCHEMBL6885410 0.82 PIN1 (0.60) PIN1ERCC1FEN1ERCC4ATM
SCHEMBL6883225 0.81 PIN1 (0.40) PIN1ERCC1FEN1ERCC4ATM
SCHEMBL6883583 0.79 ERCC1 (0.44) PIN1ERCC1FEN1ERCC4ATM
SCHEMBL6883394 0.79 EGLN1 (0.50) PIN1ERCC1FEN1ERCC4ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004096128-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-11 WO disclosed