SCHEMBL6883598

SCHEMBL6883598

COc1cccc(OC)c1-c1nc(C(=O)N(C)Cc2ccc(F)cc2)c(O)c(=O)[nH]1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TNKS O95271 1/20 0.43
TNKS2 Q9H2K2 1/20 0.43
PARP2 Q9UGN5 1/20 0.43
ERCC1 P07992 3/20 0.42
FEN1 P39748 3/20 0.42
ERCC4 Q92889 3/20 0.42
PIN1 Q13526 2/20 0.41
RXFP1 Q9HBX9 1/20 0.41
APLNR P35414 5/20 0.39
KMT2A Q03164 1/20 0.39
ATM Q13315 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6884321 0.89 HSD17B1 (0.44) TNKSTNKS2PARP2ERCC1FEN1
SCHEMBL6883583 0.89 ERCC1 (0.44) ERCC1FEN1ERCC4PIN1KMT2A
SCHEMBL6883275 0.87 RNASEH1 (0.40) TNKSERCC1FEN1ERCC4PIN1
SCHEMBL6017817 0.87 RNASEH1 (0.43) PIN1RXFP1APLNR
SCHEMBL6884446 0.87 CBFB (0.43) TNKSTNKS2PARP2ERCC1FEN1
SCHEMBL6885416 0.85 HSP90AA1 (0.41) ERCC1FEN1ERCC4PIN1RXFP1
SCHEMBL6885301 0.85 PIN1 (0.47) ERCC1FEN1ERCC4PIN1KMT2A
SCHEMBL6885410 0.83 PIN1 (0.60) ERCC1FEN1ERCC4PIN1ATM
SCHEMBL6885172 0.82 PIN1 (0.43) ERCC1FEN1ERCC4PIN1
SCHEMBL6649378 0.81 ERCC1 (0.58) TNKSTNKS2ERCC1FEN1ERCC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004096128-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-11 WO claimed
WO-2004096128-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-11 WO disclosed