SCHEMBL6889461

SCHEMBL6889461

O=C(O)c1cc(-c2cccc(CBr)c2)ccc1Cl

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACMSD Q8TDX5 4/20 0.52
PTGER1 P34995 1/20 0.49
ERCC5 P28715 1/20 0.48
FEN1 P39748 1/20 0.48
GRIK1 P39086 1/20 0.48
GRIA1 P42261 1/20 0.48
GRIA2 P42262 1/20 0.48
GRIA3 P42263 1/20 0.48
GRIA4 P48058 1/20 0.48
GRIK2 Q13002 1/20 0.48
GRIK3 Q13003 1/20 0.48
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
ALDH1A1 P00352 1/20 0.46
TP53 P04637 1/20 0.46
XDH P47989 1/20 0.45
CYP4F2 P78329 1/20 0.44
CYP4A11 Q02928 1/20 0.44
BCL2 P10415 1/20 0.44
CYP2C9 P11712 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31312276 0.86 ACMSD (0.70) ACMSDPTGER1ERCC5FEN1GRIK1
SCHEMBL31312075 0.83 CYP4F2 (0.59) ERCC5FEN1MEN1KMT2AALDH1A1
SCHEMBL787287 0.83 CYP4F2 (0.59) ERCC5FEN1MEN1KMT2AALDH1A1
SCHEMBL30402090 0.82 CYP4F2 (0.61) GRIK1GRIA1GRIA2GRIA3GRIA4
SCHEMBL844419 0.82 CYP4F2 (0.61) GRIK1GRIA1GRIA2GRIA3GRIA4
SCHEMBL122520 0.80 ACMSD (0.63) ACMSDPTGER1ERCC5FEN1GRIK1
SCHEMBL2771204 0.80 ALDH1A1 (0.68) ACMSDPTGER1ERCC5FEN1GRIK1
SCHEMBL15936129 0.79 ALDH1A1 (0.63) ACMSDERCC5FEN1GRIK1GRIA1
SCHEMBL31312218 0.78 RXRA (0.62) ACMSDERCC5FEN1GRIK1GRIA1
SCHEMBL14783994 0.76 DCLRE1B (0.57) ACMSDERCC5FEN1GRIK1GRIA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011116356-A2 POSITIVE ALLOSTERIC MODULATORS OF GROUP II MGLURS SANFORD-BURNHAM MEDICAL RESEARCH INSTITUTE (US) 2011-09-22 WO disclosed