SCHEMBL6891774

SCHEMBL6891774

CCOCC[C@H](C)NC(=O)c1cc(Cc2ccc(C(F)F)nc2)c2cccc(F)c2n1

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 3/20 0.33
POLB P06746 1/20 0.32
P2RX7 Q99572 1/20 0.32
IRAK4 Q9NWZ3 2/20 0.32
ADORA1 P30542 1/20 0.32
CHRM1 P11229 3/20 0.31
PDE1A P54750 1/20 0.31
PDE1B Q01064 1/20 0.31
PDE1C Q14123 1/20 0.31
PTGS2 P35354 1/20 0.31
MAPK1 P28482 1/20 0.31
KCNB1 Q14721 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17656783 0.76 CHRM1 (0.48) P2RX7CHRM1
SCHEMBL2223239 0.72 P2RX7 (0.33) ADORA2AP2RX7CHRM1
SCHEMBL12803022 0.72 CHRM1 (0.55) CHRM1
SCHEMBL12802494 0.72 CHRM1 (0.43) CHRM1
SCHEMBL2224850 0.67 GRM2 (0.46) ADORA2A
SCHEMBL6890674 0.66 CHRM1 (0.49) CHRM1
SCHEMBL17585463 0.66 CHRM1 (0.48) CHRM1
SCHEMBL6892942 0.65 CHRM1 (0.49) CHRM1
SCHEMBL12803346 0.65 CHRM1 (0.54) CHRM1
SCHEMBL17296540 0.64 CHRM1 (0.56) CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011084368-A1 QUINOLINE AMIDE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS MERCK SHARP & DOHME CORP. (US) 2011-07-14 WO disclosed