SCHEMBL6897446

SCHEMBL6897446

COc1cc(CC#N)cc(Br)c1O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.53
PTGS2 P35354 1/20 0.53
EGFR P00533 2/20 0.51
ALDH1A1 P00352 4/20 0.46
GAA P10253 3/20 0.46
MAPT P10636 3/20 0.46
KDM4E B2RXH2 2/20 0.46
HTT P42858 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
MEN1 O00255 4/20 0.46
KMT2A Q03164 4/20 0.46
ALOX15 P16050 3/20 0.46
ALOX12 P18054 2/20 0.46
USP2 O75604 1/20 0.46
HSD17B10 Q99714 1/20 0.46
TRPV1 Q8NER1 1/20 0.45
PTP4A3 O75365 2/20 0.41
PTP4A2 Q12974 2/20 0.41
PTP4A1 Q93096 2/20 0.41
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27936092 0.81 CA1 (0.47) PTGS2ALDH1A1GAAMAPTHTT
SCHEMBL15506125 0.80 PIK3CD (0.37) PTGS2ALDH1A1MAPTKDM4EHTT
SCHEMBL14660518 0.79 ALOX5 (0.60) ALOX5PTGS2EGFRALDH1A1GAA
SCHEMBL12766044 0.79 PTGS2 (0.60) ALOX5PTGS2EGFRALDH1A1GAA
SCHEMBL150589 0.76 MAPT (0.50) ALDH1A1GAAMAPTKDM4EHTT
SCHEMBL10345419 0.76 CA2 (0.41) ALDH1A1MAPTKDM4EHTTL3MBTL1
SCHEMBL29899617 0.76 CA2 (0.41) ALDH1A1MAPTKDM4EHTTL3MBTL1
SCHEMBL17694500 0.75 PIK3CD (0.34) PTGS2ALDH1A1MAPTKDM4EHTT
SCHEMBL1020821 0.74 PTGS2 (0.57) PTGS2MAPT
SCHEMBL9719008 0.74 ALDH1A1 (0.52) ALDH1A1GAAMAPTKDM4EHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1126833-A4 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES INC (US) 2004-09-08 EP disclosed
EP-1126833-A2 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES, INC. (US) 2001-08-29 EP disclosed
WO-2000025768-A1 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES, INC. (US) 2000-05-11 WO disclosed