SCHEMBL6902944

SCHEMBL6902944

Clc1ccc([C@H]2CCNC2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 1/20 1.00
SLC6A2 P23975 1/20 0.55
SLC6A3 Q01959 1/20 0.55
JAK3 P52333 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26690667 1.00 HTR3A (1.00) HTR3ASLC6A2SLC6A3JAK3
SCHEMBL447190 1.00 HTR3A (1.00) HTR3ASLC6A2SLC6A3JAK3
Hydrochloric Acid SCHEMBL29908691 0.98 HTR3A (0.96) HTR3ASLC6A2SLC6A3JAK3
Hydrochloric Acid SCHEMBL4573036 0.98 HTR3A (0.96) HTR3ASLC6A2SLC6A3JAK3
SCHEMBL308190 0.90 HTR3A (0.81) HTR3ASLC6A2SLC6A3
SCHEMBL16446546 0.90 HTR3A (0.81) HTR3ASLC6A2SLC6A3
SCHEMBL16446343 0.90 HTR3A (0.81) HTR3ASLC6A2SLC6A3
Oxalic Acid SCHEMBL3546578 0.89 HTR3A (0.80) HTR3AJAK3
Hydrochloric Acid SCHEMBL2884603 0.88 HTR3A (0.79) HTR3ASLC6A2SLC6A3
SCHEMBL187003 0.87 HTR3A (0.77) HTR3ASLC6A2SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4635494-A2 AMIDO HETEROAROMATIC COMPOUNDS Astrazeneca AB (SE) 2025-10-22 EP disclosed
EP-4514782-B1 AMIDO HETEROAROMATIC COMPOUNDS USEFUL IN THE TREATMENT OF LIVER DISEASES ASTRAZENECA AB (SE) 2025-09-10 EP disclosed
US-12336991-B2 Factor XIIA inhibitors UNIVERSITY OF LEEDS (GB) 2025-06-24 US disclosed
US-12291524-B2 Amido heteroaromatic compounds ASTRAZENECA AB (SE) 2025-05-06 US disclosed
EP-4514782-A1 AMIDO HETEROAROMATIC COMPOUNDS USEFUL IN THE TREATMENT OF LIVER DISEASES Astrazeneca AB (SE) 2025-03-05 EP disclosed
US-20250011311-A1 AMIDO HETEROAROMATIC COMPOUNDS ASTRAZENECA AB (SE) 2025-01-09 US disclosed
CN-119173506-A Amide heteroaromatic compounds for the treatment of liver diseases 阿斯利康(瑞典)有限公司 2024-12-20 CN disclosed
WO-2023222850-A1 AMIDO HETEROAROMATIC COMPOUNDS USEFUL IN THE TREATMENT OF LIVER DISEASES ASTRAZENECA AB (SE) 2023-11-23 WO disclosed
US-20230373983-A1 AMIDO HETEROAROMATIC COMPOUNDS ASTRAZENECA AB (SE) 2023-11-23 US disclosed
CN-111936488-B Novel compounds for the treatment of parasitic infections 葛兰素史克知识产权开发有限公司 2023-06-27 CN disclosed
US-20220305011-A1 FACTOR XIIA INHIBITORS UNIVERSITY OF LEEDS (GB) 2022-09-29 US disclosed
US-20210047299-A1 NOVEL COMPOUNDS FOR THE TREATMENT OF PARASITIC INFECTIONS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2021-02-18 US disclosed
US-20210047299-A1 NOVEL COMPOUNDS FOR THE TREATMENT OF PARASITIC INFECTIONS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2021-02-18 US disclosed
EP-3743419-A1 NOVEL COMPOUNDS FOR THE TREATMENT OF PARASITIC INFECTIONS GlaxoSmithKline Intellectual Property Development Limited (GB) 2020-12-02 EP disclosed
CN-111936488-A Novel compounds for the treatment of parasitic infections 葛兰素史克知识产权开发有限公司 2020-11-13 CN disclosed
WO-2019145360-A1 NOVEL COMPOUNDS FOR THE TREATMENT OF PARASITIC INFECTIONS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2019-08-01 WO disclosed
WO-2019145360-A1 NOVEL COMPOUNDS FOR THE TREATMENT OF PARASITIC INFECTIONS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2019-08-01 WO disclosed
EP-2681215-B1 SERINE/THREONINE KINASE INHIBITORS ARRAY BIOPHARMA INC (US) 2015-04-22 EP disclosed
WO-2011073160-A1 PYRROLIDINE DERIVATIVES AS NK - 3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2011-06-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12291524-B2 Amido heteroaromatic compounds CYP7A1, SLC10A1, CYP11B2 HTR3A 1944/4885SLC6A2 1160/4885SLC6A3 2143/4885
US-20210047299-A1 NOVEL COMPOUNDS FOR THE TREATMENT OF PARASITIC INFECTIONS PIGO, ENPP2, THPO HTR3A 4719/4885SLC6A2 2997/4885SLC6A3 3645/4885
US-20230373983-A1 AMIDO HETEROAROMATIC COMPOUNDS CYP7A1, SLC10A1, CYP11B2 HTR3A 1944/4885SLC6A2 1160/4885SLC6A3 2143/4885
US-20220305011-A1 FACTOR XIIA INHIBITORS F11, F13B, F12 HTR3A 4363/4885SLC6A2 4224/4885SLC6A3 4773/4885
US-12336991-B2 Factor XIIA inhibitors F11, F13B, F12 HTR3A 4363/4885SLC6A2 4224/4885SLC6A3 4773/4885
US-20250011311-A1 AMIDO HETEROAROMATIC COMPOUNDS CYP7A1, SLC10A1, CYP11B2 HTR3A 1944/4885SLC6A2 1160/4885SLC6A3 2143/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.