SCHEMBL447190

SCHEMBL447190

Clc1ccc(C2CCNC2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 1/20 1.00
SLC6A2 P23975 1/20 0.55
SLC6A3 Q01959 1/20 0.55
JAK3 P52333 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6902944 1.00 HTR3A (1.00) HTR3ASLC6A2SLC6A3JAK3
SCHEMBL26690667 1.00 HTR3A (1.00) HTR3ASLC6A2SLC6A3JAK3
Hydrochloric Acid SCHEMBL29908691 0.98 HTR3A (0.96) HTR3ASLC6A2SLC6A3JAK3
Hydrochloric Acid SCHEMBL4573036 0.98 HTR3A (0.96) HTR3ASLC6A2SLC6A3JAK3
SCHEMBL308190 0.90 HTR3A (0.81) HTR3ASLC6A2SLC6A3
SCHEMBL16446546 0.90 HTR3A (0.81) HTR3ASLC6A2SLC6A3
SCHEMBL16446343 0.90 HTR3A (0.81) HTR3ASLC6A2SLC6A3
Oxalic Acid SCHEMBL3546578 0.89 HTR3A (0.80) HTR3AJAK3
Hydrochloric Acid SCHEMBL2884603 0.88 HTR3A (0.79) HTR3ASLC6A2SLC6A3
SCHEMBL187003 0.87 HTR3A (0.77) HTR3ASLC6A2SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 184 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10792262-B1 Stabilized formulations of 4-amino-3-substituted butanoic acid derivatives SAOL INTERNATIONAL LIMITED (BM) 2020-10-06 US claimed
US-10751312-B1 2020-08-25 US claimed
EP-4635494-A2 AMIDO HETEROAROMATIC COMPOUNDS Astrazeneca AB (SE) 2025-10-22 EP disclosed
EP-4514782-B1 AMIDO HETEROAROMATIC COMPOUNDS USEFUL IN THE TREATMENT OF LIVER DISEASES ASTRAZENECA AB (SE) 2025-09-10 EP disclosed
US-12291524-B2 Amido heteroaromatic compounds ASTRAZENECA AB (SE) 2025-05-06 US disclosed
WO-2025045746-A1 PYRAZOLE DERIVATIVES AS SARM1 INHIBITORS USEFUL FOR THE TREATMENT OF NEURODEGENERATIVE DISORDERS F. HOFFMANN-LA ROCHE AG (CH) 2025-03-06 WO disclosed
EP-4514782-A1 AMIDO HETEROAROMATIC COMPOUNDS USEFUL IN THE TREATMENT OF LIVER DISEASES Astrazeneca AB (SE) 2025-03-05 EP disclosed
US-20250011311-A1 AMIDO HETEROAROMATIC COMPOUNDS ASTRAZENECA AB (SE) 2025-01-09 US disclosed
US-20240408042-A1 ORALLY DISINTEGRATING BACLOFEN COMPOSITIONS AND METHODS OF MAKING SAME CLINICAL RES ASSOCIATES LLC (US) 2024-12-12 US disclosed
CN-114072398-B Compounds that inhibit TDG activity 上海仕谱生物科技有限公司 2024-06-11 CN disclosed
US-11931328-B2 Stabilized formulations of 4-amino-3-substituted butanoic acid derivatives AMNEAL PHARMACEUTICALS LLC (US) 2024-03-19 US disclosed
WO-2005019163-A2 ACYLOXYALKYL CARBAMATE PRODRUGS, METHODS OF SYNTHESIS AND USE XENOPORT, INC. (US) 2005-03-03 WO disclosed
CN-1150165-C 1-arylsulfonyl-2-aryl-pyrrolidine derivatives for the treatment of central nervous system disorders - 2004-05-19 CN disclosed
CN-1345311-A 1-arenesulfonyl-2-aryl-pyrolidine and piperidine derivatives for treatment of CNS disorders HOFFMANN LA ROCHE (CH) 2002-04-17 CN disclosed
EP-0920425-A1 SUBSTITUTED 4-(1H-BENZIMIDAZOL-2-YL-AMINO)PIPERIDINES USEFUL FOR THE TREATMENT OF ALLERGIC DISEASES HOECHST MARION ROUSSEL, INC. (US) 1999-06-09 EP disclosed
US-5824690-A TREATING ASTHMA, COUGH HOECHST MARION ROUSSEL INC. (US) 1998-10-20 US disclosed
WO-1997019074-A1 SUBSTITUTED 4-(1H-BENZIMIDAZOL-2-YL-AMINO)PIPERIDINES USEFUL FOR THE TREATMENT OF ALLERGIC DISEASES HOECHST MARION ROUSSEL, INC. (US) 1997-05-29 WO disclosed
EP-0272208-B1 AROMATICALLY SUBSTITUTED AZACYCLO-ALKYLALKANEDIPHOSPHONIC ACIDS CIBA-GEIGY AG (CH) 1991-06-12 EP disclosed
US-4871720-A Aromatically substituted azacycloalkyl-alkanediphosphonic acids useful for the treatment of illnesses that can be attributed to calcium metabolism disorders CIBA-GEIGY CORPORATION (US) 1989-10-03 US disclosed
EP-0272208-A1 Aromatically substituted azacyclo-alkylalkanediphosphonic acids CIBA-GEIGY AG (CH) 1988-06-22 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10792262-B1 Stabilized formulations of 4-amino-3-substituted butanoic acid derivatives ABAT, GABRA6, BCAT2 HTR3A 106/4885SLC6A2 1837/4885SLC6A3 1431/4885
US-12291524-B2 Amido heteroaromatic compounds CYP7A1, SLC10A1, CYP11B2 HTR3A 1944/4885SLC6A2 1160/4885SLC6A3 2143/4885
US-20240408042-A1 ORALLY DISINTEGRATING BACLOFEN COMPOSITIONS AND METHODS OF MAKING SAME GABBR2, GABBR1, GABRB2 HTR3A 1318/4885SLC6A2 587/4885SLC6A3 796/4885
US-11931328-B2 Stabilized formulations of 4-amino-3-substituted butanoic acid derivatives GABRA6, GABBR1, GABBR2 HTR3A 75/4885SLC6A2 908/4885SLC6A3 1046/4885
US-10751312-B1 LIPA, CEL, GANC HTR3A 4252/4885SLC6A2 4437/4885SLC6A3 4714/4885
US-20250011311-A1 AMIDO HETEROAROMATIC COMPOUNDS CYP7A1, SLC10A1, CYP11B2 HTR3A 1944/4885SLC6A2 1160/4885SLC6A3 2143/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.