SCHEMBL690438

SCHEMBL690438

C=C(CC(OCC)(OCC)Oc1ccccc1)C(=O)O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 4/20 0.36
MAPT P10636 3/20 0.36
ALDH1A1 P00352 1/20 0.36
TET2 Q6N021 1/20 0.35
METAP2 P50579 1/20 0.34
METAP1 P53582 1/20 0.34
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
HPGD P15428 1/20 0.33
CRHBP P24387 1/20 0.33
CRHR2 Q13324 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
KDM4E B2RXH2 1/20 0.33
PIN1 Q13526 1/20 0.33
ALOX15 P16050 1/20 0.33
LMNA P02545 1/20 0.32
GAA P10253 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
EGFR P00533 1/20 0.32
PPARA Q07869 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18225556 0.86 LMNA (0.31) ALDH1A1LMNA
SCHEMBL9290995 0.76 MAPT (0.38) PPARGMAPTALDH1A1NPC1RAB9A
SCHEMBL691683 0.75 TDP1 (0.40) MAPTALDH1A1NPC1RAB9AHPGD
SCHEMBL11228920 0.75 LTA4H (0.38) PPARGMAPTALDH1A1NPC1RAB9A
SCHEMBL690076 0.74 AKR1C3 (0.37) PPARGMAPTALDH1A1NPC1RAB9A
SCHEMBL690077 0.74 AKR1C3 (0.37) PPARGMAPTALDH1A1NPC1RAB9A
SCHEMBL691151 0.72 THRB (0.49) MAPTALDH1A1NPC1RAB9AHPGD
SCHEMBL9820438 0.70 THRB (0.40) MAPTALDH1A1NPC1RAB9ALMNA
SCHEMBL10385264 0.69 PPARG (0.42) PPARGMAPTNPC1RAB9AHPGD
SCHEMBL28377681 0.69 ALOX15 (0.48) PPARGALOX15PPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9907881-B2 Crosslinked, hydrophobic acrylic copolymer made of 2-phenoxytetraethylene-glycol acrylate and intended for intraocular lenses ACRYLIAN (FR) 2018-03-06 US claimed
EP-3110464-B1 CROSSLINKED, HYDROPHOBIC ACRYLIC COPOLYMER MADE OF 2-PHENOXY-TETRAETHYLENE-GLYCOL ACRYLATE AND INTENDED FOR INTRAOCULAR LENSES ACRYLIAN (FR) 2017-11-01 EP claimed
EP-3110464-A1 CROSSLINKED, HYDROPHOBIC ACRYLIC COPOLYMER MADE OF 2-PHENOXY-TETRAETHYLENE-GLYCOL ACRYLATE AND INTENDED FOR INTRAOCULAR LENSES Acrylian (FR) 2017-01-04 EP claimed
WO-2015128555-A1 CROSSLINKED, HYDROPHOBIC ACRYLIC COPOLYMER MADE OF 2-PHENOXY-TETRAETHYLENE-GLYCOL ACRYLATE AND INTENDED FOR INTRAOCULAR LENSES ACRYLIAN (FR) 2015-09-03 WO claimed
EP-2285427-B1 HYDROPHOBIC ACRYLIC POLYMER MATERIAL FOR AN INTRAOCULAR LENS, HAVING AN ENHANCED FLEXIBILITY DUE TO THE USE OF A TRANSFER AGENT ACRYLIAN (FR) 2012-02-29 EP claimed
EP-2285427-A1 HYDROPHOBIC ACRYLIC POLYMER MATERIAL FOR AN INTRAOCULAR LENS, HAVING AN ENHANCED FLEXIBILITY DUE TO THE USE OF A TRANSFER AGENT Acrylian (FR) 2011-02-23 EP claimed
WO-2009138591-A1 HYDROPHOBIC ACRYLIC POLYMER MATERIAL FOR AN INTRAOCULAR LENS, HAVING AN ENHANCED FLEXIBILITY DUE TO THE USE OF A TRANSFER AGENT ACRYLIAN (FR) 2009-11-19 WO claimed
US-9907881-B2 Crosslinked, hydrophobic acrylic copolymer made of 2-phenoxytetraethylene-glycol acrylate and intended for intraocular lenses ACRYLIAN (FR) 2018-03-06 US disclosed
EP-3110464-B1 CROSSLINKED, HYDROPHOBIC ACRYLIC COPOLYMER MADE OF 2-PHENOXY-TETRAETHYLENE-GLYCOL ACRYLATE AND INTENDED FOR INTRAOCULAR LENSES ACRYLIAN (FR) 2017-11-01 EP disclosed
EP-3110464-A1 CROSSLINKED, HYDROPHOBIC ACRYLIC COPOLYMER MADE OF 2-PHENOXY-TETRAETHYLENE-GLYCOL ACRYLATE AND INTENDED FOR INTRAOCULAR LENSES Acrylian (FR) 2017-01-04 EP disclosed
US-20160331864-A1 CROSSLINKED, HYDROPHOBIC ACRYLIC COPOLYMER MADE OF 2- PHENOXYTETRAETHYLENE-GLYCOL ACRYLATE AND INTENDED FOR INTRAOCULAR LENSES ACRYLIAN (FR) 2016-11-17 US disclosed
WO-2015128555-A1 CROSSLINKED, HYDROPHOBIC ACRYLIC COPOLYMER MADE OF 2-PHENOXY-TETRAETHYLENE-GLYCOL ACRYLATE AND INTENDED FOR INTRAOCULAR LENSES ACRYLIAN (FR) 2015-09-03 WO disclosed
EP-2285427-B1 HYDROPHOBIC ACRYLIC POLYMER MATERIAL FOR AN INTRAOCULAR LENS, HAVING AN ENHANCED FLEXIBILITY DUE TO THE USE OF A TRANSFER AGENT ACRYLIAN (FR) 2012-02-29 EP disclosed
EP-2285427-A1 HYDROPHOBIC ACRYLIC POLYMER MATERIAL FOR AN INTRAOCULAR LENS, HAVING AN ENHANCED FLEXIBILITY DUE TO THE USE OF A TRANSFER AGENT Acrylian (FR) 2011-02-23 EP disclosed
WO-2009138591-A1 HYDROPHOBIC ACRYLIC POLYMER MATERIAL FOR AN INTRAOCULAR LENS, HAVING AN ENHANCED FLEXIBILITY DUE TO THE USE OF A TRANSFER AGENT ACRYLIAN (FR) 2009-11-19 WO disclosed