SCHEMBL6906283

SCHEMBL6906283

CN(Cc1ccc(C(C)(C)C)cc1)Cc1ccccc1Br

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 4/20 0.65
LMNA P02545 3/20 0.65
SIGMAR1 Q99720 2/20 0.65
ACHE P22303 2/20 0.65
KCNH2 Q12809 2/20 0.65
NR1I2 O75469 1/20 0.65
ADRA2A P08913 1/20 0.65
SLC6A2 P23975 1/20 0.65
HTR2A P28223 1/20 0.65
SLC6A4 P31645 1/20 0.65
PYCR1 P32322 2/20 0.50
CYP1A2 P05177 3/20 0.45
CYP2C19 P33261 3/20 0.45
CYP2C9 P11712 1/20 0.45
HIF1A Q16665 1/20 0.45
TSHR P16473 2/20 0.41
TMEM97 Q5BJF2 1/20 0.41
TAAR1 Q96RJ0 1/20 0.41
CYP19A1 P11511 2/20 0.40
KDM4E B2RXH2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6914436 0.87 CYP2D6 (0.60) CYP2D6LMNASIGMAR1ACHEKCNH2
SCHEMBL9722145 0.82 CYP2D6 (0.67) CYP2D6LMNASIGMAR1ACHEKCNH2
Butenafine SCHEMBL29354083 0.79 CYP2D6 (1.00) CYP2D6LMNASIGMAR1ACHEKCNH2
SCHEMBL8041553 0.79 TACR1 (0.63) CYP2D6LMNASIGMAR1ACHEKCNH2
Butenafine SCHEMBL65526 0.79 CYP2D6 (1.00) CYP2D6LMNASIGMAR1ACHEKCNH2
Butenafine SCHEMBL20456391 0.79 CYP2D6 (1.00) CYP2D6LMNASIGMAR1ACHEKCNH2
Butenafine SCHEMBL262301 0.78 LMNA (0.97) CYP2D6LMNASIGMAR1ACHEKCNH2
Butenafine SCHEMBL676912 0.78 LMNA (0.97) CYP2D6LMNASIGMAR1ACHEKCNH2
Butenafine SCHEMBL29459249 0.78 LMNA (0.97) CYP2D6LMNASIGMAR1ACHEKCNH2
SCHEMBL6914321 0.78 SIGMAR1 (0.50) CYP2D6LMNASIGMAR1ACHEKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1112998-B1 AMINE DERIVATIVES POLA CHEM IND INC (JP) 2004-12-08 EP disclosed
US-6586633-B1 Antifungal agents POLA CHEMICAL INDUSTRIES, INC. (JP) 2003-07-01 US disclosed
EP-1112998-A1 AMINE DERIVATIVES POLA CHEMICAL INDUSTRIES, INC. (JP) 2001-07-04 EP disclosed