SCHEMBL6907289

SCHEMBL6907289

Nc1cccc(-n2[nH]c3c(c2=O)CN(Cc2cccnc2)CC3)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.43
GABRA3 P34903 1/20 0.43
GABRA2 P47869 1/20 0.43
CLPP Q16740 1/20 0.42
KDM4E B2RXH2 2/20 0.41
GFER P55789 1/20 0.41
DRD2 P14416 1/20 0.41
KCNH2 Q12809 1/20 0.41
POLB P06746 1/20 0.41
CYBB P04839 3/20 0.40
NOX4 Q9NPH5 3/20 0.40
NOX5 Q96PH1 2/20 0.40
NOX1 Q9Y5S8 2/20 0.40
COMT P21964 1/20 0.40
CYP17A1 P05093 2/20 0.39
CYP3A4 P08684 2/20 0.39
CHRNB2 P17787 1/20 0.39
CHRNA4 P43681 1/20 0.39
OPRM1 P35372 1/20 0.39
OPRD1 P41143 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6910467 0.92 COMT (0.42) GABRA1GABRA3GABRA2CLPPKDM4E
SCHEMBL2301876 0.88 CLPP (0.50) GABRA1GABRA3GABRA2CLPPCYBB
SCHEMBL2305199 0.86 CLPP (0.44) GABRA1GABRA3GABRA2CLPPCYBB
SCHEMBL6908946 0.85 CLPP (0.37) CLPPKDM4ECHRNB2CHRNA4
SCHEMBL6907625 0.84 CLPP (0.42) CLPPKDM4EDRD2
SCHEMBL2302142 0.83 CLPP (0.48) GABRA1GABRA3GABRA2CLPPCYBB
SCHEMBL2302100 0.83 KDM4E (0.43) GABRA1GABRA3GABRA2CLPPKDM4E
SCHEMBL6909785 0.82 BRS3 (0.44) CLPPKDM4EDRD2KCNH2POLB
SCHEMBL6911739 0.81 SLC6A5 (0.42) CLPPDRD2
SCHEMBL6909385 0.79 CLPP (0.40) GABRA1GABRA2CLPPKCNH2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011101804-A1 PYRAZOLO PIPERIDINE DERIVATIVES AS NADPH OXIDASE INHIBITORS GENKYOTEX SA (CH) 2011-08-25 WO disclosed