SCHEMBL6908503

SCHEMBL6908503

Nc1ccc(CN2CCc3[nH]n(Cc4ccccc4)c(=O)c3C2)cc1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACHE P22303 3/20 0.48
SLC6A5 Q9Y345 1/20 0.47
AKR1B1 P15121 1/20 0.45
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
GABRA1 P14867 1/20 0.43
GABRA2 P47869 1/20 0.43
CLPP Q16740 4/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
CYP1A2 P05177 1/20 0.43
GAA P10253 1/20 0.43
CYP2C9 P11712 1/20 0.43
ADORA2A P29274 1/20 0.43
BRS3 P32247 1/20 0.42
PNMT P11086 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2301297 0.93 ACHE (0.54) ACHESLC6A5AKR1B1GABRA1GABRA2
SCHEMBL6908510 0.90 ACHE (0.46) ACHESLC6A5AKR1B1MEN1KMT2A
SCHEMBL2299422 0.89 CLPP (0.53) ACHESLC6A5AKR1B1GABRA1GABRA2
SCHEMBL2300918 0.89 CLPP (0.53) ACHESLC6A5AKR1B1GABRA1GABRA2
SCHEMBL2310779 0.85 CLPP (0.46) ACHESLC6A5AKR1B1MEN1KMT2A
SCHEMBL2301137 0.85 SIGMAR1 (0.53) ACHESLC6A5AKR1B1MEN1KMT2A
SCHEMBL2303283 0.85 ACHE (0.56) ACHEKMT2AGABRA1GABRA2CLPP
SCHEMBL6907424 0.85 ALDH1A1 (0.42) ACHESLC6A5AKR1B1MEN1KMT2A
SCHEMBL2339909 0.85 ACHE (0.47) ACHESLC6A5AKR1B1MEN1KMT2A
SCHEMBL6907587 0.84 ALDH1A1 (0.49) ACHESLC6A5CLPPKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011101804-A1 PYRAZOLO PIPERIDINE DERIVATIVES AS NADPH OXIDASE INHIBITORS GENKYOTEX SA (CH) 2011-08-25 WO disclosed