SCHEMBL6911686

SCHEMBL6911686

Nc1cccc(-n2[nH]c3c(c2=O)CCN(Cc2cccc(Cl)c2)C3)c1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.51
GAA P10253 1/20 0.51
KMT2A Q03164 1/20 0.51
ATM Q13315 1/20 0.51
CLPP Q16740 5/20 0.42
DRD2 P14416 1/20 0.42
DRD4 P21917 1/20 0.42
DRD3 P35462 1/20 0.42
SLC6A5 Q9Y345 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
CYBB P04839 2/20 0.41
NOX5 Q96PH1 2/20 0.41
NOX4 Q9NPH5 2/20 0.41
NOX1 Q9Y5S8 2/20 0.41
TRPV1 Q8NER1 1/20 0.40
MAPT P10636 2/20 0.40
TSHR P16473 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6911739 0.93 SLC6A5 (0.42) MEN1GAAKMT2AATMCLPP
SCHEMBL2352634 0.90 MEN1 (0.54) MEN1GAAKMT2AATMCLPP
SCHEMBL6911338 0.89 MEN1 (0.44) MEN1GAAKMT2AATMCLPP
SCHEMBL2343325 0.88 MEN1 (0.54) MEN1GAAKMT2AATMCLPP
SCHEMBL2350571 0.86 DRD2 (0.55) MEN1GAAKMT2AATMCLPP
SCHEMBL2347778 0.85 CLPP (0.49) MEN1GAAKMT2AATMCLPP
SCHEMBL6911024 0.85 BRS3 (0.44) GAACLPPDRD2DRD3SLC6A5
SCHEMBL6910461 0.85 MEN1 (0.37) MEN1GAAKMT2AATMCLPP
SCHEMBL6910467 0.84 COMT (0.42) CLPPDRD2CYBBNOX5NOX4
SCHEMBL6907625 0.84 CLPP (0.42) MEN1KMT2ACLPPDRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011101805-A1 PYRAZOLO PIPERIDINE DERIVATIVES AS NADPH OXIDASE INHIBITORS GENKYOTEX SA (CH) 2011-08-25 WO disclosed