SCHEMBL6921671

SCHEMBL6921671

CCCOC1CCN(CC(=O)c2cc(C)n(-c3ccc(N)cc3)c2C)CC1

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 7/20 0.58
RAB9A P51151 5/20 0.58
NPC1 O15118 4/20 0.58
USP14 P54578 9/20 0.55
USP7 Q93009 3/20 0.55
USP5 P45974 2/20 0.55
HPGD P15428 3/20 0.54
KDM4E B2RXH2 3/20 0.53
POLB P06746 1/20 0.53
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
MAPT P10636 1/20 0.46
ALDH1A1 P00352 1/20 0.46
HTT P42858 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19749176 0.92 SMN1; SMN2 (0.65) SMN1; SMN2RAB9ANPC1USP14USP7
SCHEMBL19749206 0.90 SMN1; SMN2 (0.58) SMN1; SMN2RAB9ANPC1USP14USP7
SCHEMBL17949714 0.90 SMN1; SMN2 (0.68) SMN1; SMN2RAB9ANPC1USP14USP7
SCHEMBL6922889 0.88 SMN1; SMN2 (0.62) SMN1; SMN2RAB9ANPC1USP14USP7
SCHEMBL6922433 0.85 SMN1; SMN2 (0.59) SMN1; SMN2RAB9ANPC1USP14USP7
SCHEMBL6923174 0.84 SMN1; SMN2 (0.63) SMN1; SMN2RAB9ANPC1USP14USP7
SCHEMBL6923200 0.84 SMN1; SMN2 (0.79) SMN1; SMN2RAB9ANPC1USP14USP7
SCHEMBL6923352 0.84 SMN1; SMN2 (0.57) SMN1; SMN2RAB9ANPC1USP14USP7
SCHEMBL6921573 0.81 SMN1; SMN2 (0.62) SMN1; SMN2RAB9ANPC1USP14USP7
SCHEMBL19501668 0.81 KDM4E (0.45) SMN1; SMN2RAB9ANPC1USP14USP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160214989-A1 Compositions and Methods for Enhancing Proteasome Activity THE ASSAY DEPOT, INC. 2016-07-28 US disclosed
US-20150335652-A1 USP14 Inhibitors for Treating or Preventing Viral Infections PRESIDENT AND FELLOWS OF HARVARD COLLEGE 2015-11-26 US disclosed
US-20140275169-A1 Combination Therapies for Enhancing Protein Degradation THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2014-09-18 US disclosed
WO-2014116228-A1 USP14 INHIBITORS FOR TREATING OR PREVENTING VIRAL INFECTIONS PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2014-07-31 WO disclosed
US-20130045992-A1 Compositions and Methods for Enhancing Proteasome Activity PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2013-02-21 US disclosed
WO-2011094545-A2 COMPOSITIONS AND METHODS FOR ENHANCING PROTEASOME ACTIVITY PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2011-08-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150335652-A1 USP14 Inhibitors for Treating or Preventing Viral Infections USP14, USP1, USP13 SMN1; SMN2 1593/4885RAB9A 1746/4885NPC1 813/4885
US-20130045992-A1 Compositions and Methods for Enhancing Proteasome Activity PSMG3, PSMB11, PSME3 SMN1; SMN2 307/4885RAB9A 2464/4885NPC1 2654/4885
US-20160214989-A1 Compositions and Methods for Enhancing Proteasome Activity PSMG3, PSME3, PSMB11 SMN1; SMN2 307/4885RAB9A 2509/4885NPC1 2643/4885
US-20140275169-A1 Combination Therapies for Enhancing Protein Degradation HSPA2, HSPBP1, HSPH1 SMN1; SMN2 544/4885RAB9A 4241/4885NPC1 3460/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.