SCHEMBL6926972

SCHEMBL6926972

CC(=O)Nc1ccc(C(=O)COC(C)=O)cn1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.50
PTK2 Q05397 1/20 0.50
CYP1A2 P05177 1/20 0.46
GAA P10253 1/20 0.46
GRIN2B Q13224 1/20 0.45
HCAR3 P49019 2/20 0.44
RAB9A P51151 5/20 0.42
MAPT P10636 3/20 0.42
HSD17B10 Q99714 2/20 0.42
HTT P42858 1/20 0.42
NPC1 O15118 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.40
KMT2A Q03164 1/20 0.40
KDM4E B2RXH2 1/20 0.40
TP53 P04637 1/20 0.40
HPGD P15428 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6920233 0.86 PTK2 (0.46) ALDH1A1PTK2CYP1A2GAAGRIN2B
SCHEMBL6924749 0.85 RAB9A (0.56) PTK2GAAGRIN2BHCAR3RAB9A
SCHEMBL16463469 0.81 PTK2 (0.56) PTK2CYP1A2GAAGRIN2BHCAR3
SCHEMBL6923544 0.81 PTK2 (0.56) PTK2CYP1A2GAAGRIN2BHCAR3
SCHEMBL1203341 0.80 PTK2 (0.54) PTK2CYP1A2GAAGRIN2BHCAR3
SCHEMBL6576391 0.80 ALDH1A1 (0.58) ALDH1A1PTK2CYP1A2GAAGRIN2B
SCHEMBL16463731 0.79 PTK2 (0.53) PTK2CYP1A2GAAGRIN2BHCAR3
SCHEMBL7093993 0.77 PTK2 (0.62) PTK2CYP1A2GAAHCAR3RAB9A
SCHEMBL1854705 0.76 MAPK1 (0.59) ALDH1A1PTK2CYP1A2GAAHCAR3
SCHEMBL82675 0.76 HCAR3 (0.68) PTK2CYP1A2GAAHCAR3KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6642387-B2 Dehalogenation esterification; efficient; no toxic materials KANEKA CORPORATION (JP) 2003-11-04 US disclosed
US-20030130521-A1 Substituted acetylpyridine derivatives and process for the preparation of intermediates for optically active beta3 agonist by the use of the same KANEKA CORPORATION (JP) 2003-07-10 US disclosed
US-6515134-B1 A production method of an optically active hydroxyethyl pyridine derivative represented by the general formula which comprises using a microorganism-derived carbonyl reducing enzyme or a culture of a microorganism having an ability of KANEKA CORPORATION (JP) 2003-02-04 US disclosed
EP-1153919-A1 SUBSTITUTED ACETYLPYRIDINE DERIVATIVES AND PROCESS FOR THE PREPARATION OF INTERMEDIATES FOR OPTICALLY ACTIVE BETA3 AGONIST BY THE USE OF THE SAME KANEKA CORPORATION (JP) 2001-11-14 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030130521-A1 Substituted acetylpyridine derivatives and process for the preparation of intermediates for optically active beta3 agonist by the use of the same ADRB3, ADRB2, ADRB1 ALDH1A1 184/4885PTK2 3057/4885CYP1A2 138/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.