SCHEMBL6927610

SCHEMBL6927610

CC(=O)N(C#N)Cc1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.52
TSPO P30536 1/20 0.46
NPC1 O15118 3/20 0.46
RAB9A P51151 2/20 0.46
CA12 O43570 1/20 0.46
CA9 Q16790 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.45
CRHBP P24387 1/20 0.45
CRHR2 Q13324 1/20 0.45
LMNA P02545 1/20 0.44
POLB P06746 1/20 0.44
CTSL P07711 2/20 0.43
CTSS P25774 2/20 0.43
ALOX5 P09917 1/20 0.43
PTGS1 P23219 1/20 0.43
PTGS2 P35354 1/20 0.43
KMT2A Q03164 3/20 0.42
MEN1 O00255 2/20 0.42
TSHR P16473 1/20 0.42
CTSB P07858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10628165 0.90 ALDH1A1 (0.40) ALDH1A1TSPORAB9AL3MBTL1CRHBP
SCHEMBL16179158 0.86 ALDH1A1 (0.57) ALDH1A1NPC1RAB9ACA12CA9
SCHEMBL3250775 0.83 TSPO (0.47) ALDH1A1TSPONPC1RAB9ACA12
SCHEMBL3457762 0.82 ALDH1A1 (0.47) ALDH1A1NPC1RAB9AALOX5KMT2A
SCHEMBL3245208 0.81 TSPO (0.46) ALDH1A1TSPONPC1RAB9ACA12
SCHEMBL23805069 0.81 ALDH1A1 (0.52) ALDH1A1NPC1RAB9ACA12CA9
SCHEMBL5373794 0.80 ALOX5 (0.47) ALDH1A1NPC1RAB9ALMNAALOX5
SCHEMBL10630145 0.79 ALOX5 (0.50) ALDH1A1NPC1RAB9AL3MBTL1LMNA
SCHEMBL7919193 0.77 TSHR (0.45) ALDH1A1TSPOL3MBTL1CRHBPCRHR2
SCHEMBL7919236 0.76 LMNA (0.51) ALDH1A1TSPONPC1LMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3262110-B1 IMPREGNATING RESINS WHICH ARE STABLE WHEN STORED AND ELECTRO ISOLATION TAPES SIEMENS ENERGY GLOBAL GMBH & CO KG (DE) 2023-03-29 EP disclosed
CN-107580615-B Storage-stable impregnating resin and electrical insulating tape 西门子公司 2020-07-21 CN disclosed
US-10479857-B2 Storage-stable impregnating resins and electrical insulating tapes SIEMENS AKTIENGESELLSCHAFT (DE) 2019-11-19 US disclosed
US-20180171066-A1 STORAGE-STABLE IMPREGNATING RESINS AND ELECTRICAL INSULATING TAPES SIEMENS AKTIENGESELLSCHAFT (DE) 2018-06-21 US disclosed
EP-3262110-A1 STORAGE-STABLE IMPREGNATING RESINS AND ELECTRICAL INSULATING TAPES Siemens Aktiengesellschaft (DE) 2018-01-03 EP disclosed
WO-2016180595-A1 STORAGE-STABLE IMPREGNATING RESINS AND ELECTRICAL INSULATING TAPES SIEMENS AKTIENGESELLSCHAFT (DE) 2016-11-17 WO disclosed
EP-3091049-A1 IMPREGNATING RESINS WHICH ARE STABLE WHEN STORED AND ELECTRO ISOLATION TAPES Siemens Aktiengesellschaft (DE) 2016-11-09 EP disclosed
EP-1161417-B1 METHODS AND COMPOSITIONS FOR TREATING LEUKEMIA HSC RES DEV LP (CA) 2003-12-03 EP disclosed
EP-1161417-A1 METHODS AND COMPOSITIONS FOR TREATING LEUKEMIA HSC Research and Development Limited Partnership (CA) 2001-12-12 EP disclosed
WO-2000055128-A1 METHODS AND COMPOSITIONS FOR TREATING LEUKEMIA HSC RESEARCH AND DEVELOPMENT LIMITED PARTNERSHIP (CA) 2000-09-21 WO disclosed
EP-0087393-B1 PROCESS FOR THE PREPARATION OF ISOMELAMINES, AND THEIR USE CIBA-GEIGY AG (CH) 1987-01-14 EP disclosed
EP-0087394-B1 PROCESS FOR THE PREPARATION OF N-SUBSTITUTED N-CYANO-AMIDES AND THEIR USE CIBA-GEIGY AG (CH) 1986-05-14 EP disclosed
US-4550203-A REACTING AMIDE SALT WITH ALKYLATING AGENT CIBA GEIGY CORPORATION (US) 1985-10-29 US disclosed
US-4537946-A POLYEDOXIDE CURING AGENTS CIBA-GEIGY CORPORATION (US) 1985-08-27 US disclosed
US-4499268-A REACTING N-CYANO-N-(AR OR CYCLO)ALKYLCARBOXLIC AMINE WITH EITHER SODIUM(OR POTASSIUM) HYDROXIDE), AMINE, OR ALCOHOL CIBA GEIGY CORPORATION (US) 1985-02-12 US disclosed
EP-0087394-A2 Process for the preparation of N-substituted N-cyano-amides and their use CIBA-GEIGY AG (CH) 1983-08-31 EP disclosed
EP-0087393-A2 Process for the preparation of isomelamines, and their use CIBA-GEIGY AG (CH) 1983-08-31 EP disclosed