SCHEMBL6929002

SCHEMBL6929002

COC(C(=O)O)c1ccc2ccccc2c1C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NCEH1 Q6PIU2 1/20 0.43
CYP1A2 P05177 1/20 0.42
CYP2A6 P11509 1/20 0.42
TSHR P16473 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.40
KDM4E B2RXH2 2/20 0.40
HPGD P15428 1/20 0.40
AKR1B1 P15121 2/20 0.38
WDR5 P61964 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
FABP4 P15090 1/20 0.37
FABP5 Q01469 1/20 0.37
ALDH1A1 P00352 2/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
PPARG P37231 2/20 0.37
PPARA Q07869 2/20 0.37
PKM P14618 1/20 0.37
LDHA P00338 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8728993 0.82 ALDH1A1 (0.45) CYP1A2KDM4EHPGDFABP4FABP5
SCHEMBL11460736 0.80 AKR1B1 (0.53) NCEH1CYP1A2CYP2A6TSHRL3MBTL1
SCHEMBL10830584 0.78 ALDH1A1 (0.43) NCEH1CYP1A2CYP2A6TSHRL3MBTL1
SCHEMBL11556826 0.75 FABP4 (0.49) TSHRL3MBTL1KDM4EHPGDFABP4
Hydrogen Peroxide SCHEMBL8610670 0.74 TSHR (0.52) NCEH1CYP1A2CYP2A6TSHRL3MBTL1
SCHEMBL9445845 0.73 LMNA (0.45) L3MBTL1FABP4FABP5ALDH1A1PPARA
SCHEMBL9445842 0.73 LMNA (0.45) L3MBTL1FABP4FABP5ALDH1A1PPARA
SCHEMBL9445841 0.73 LMNA (0.45) L3MBTL1FABP4FABP5ALDH1A1PPARA
SCHEMBL9537762 0.73 KDM4E (0.49) KDM4EHPGDALDH1A1MEN1KMT2A
SCHEMBL6392222 0.72 ALDH1A1 (0.47) NCEH1CYP1A2KDM4EHPGDAKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1148783-A4 CONVERTING COX INHIBITION COMPOUNDS THAT ARE NOT COX-2 SELECTIVE INHIBITORS TO DERIVATIVES THAT ARE COX-2 SELECTIVE INHIBITORS UNIV VANDERBILT (US) 2003-05-21 EP claimed
EP-1148783-A1 CONVERTING COX INHIBITION COMPOUNDS THAT ARE NOT COX-2 SELECTIVE INHIBITORS TO DERIVATIVES THAT ARE COX-2 SELECTIVE INHIBITORS Vanderbilt University (US) 2001-10-31 EP claimed
WO-2000040087-A1 CONVERTING COX INHIBITION COMPOUNDS THAT ARE NOT COX-2 SELECTIVE INHIBITORS TO DERIVATIVES THAT ARE COX-2 SELECTIVE INHIBITORS VANDERBILT UNIVERSITY (US) 2000-07-13 WO claimed
US-4565877-A Naphthalene derivatives and method for preparation thereof TANABE SEIYAKU CO., LTD. (JP) 1986-01-21 US disclosed
EP-0107149-B1 NOVEL NAPHTHALENE DERIVATIVES AND METHOD FOR PREPARATION THEREOF Tanabe Seiyaku Co., Ltd. (JP) 1985-10-16 EP disclosed