SCHEMBL6932616

SCHEMBL6932616

CN1CCN(c2ccc(C(N)=O)c3c2CC(NC(=O)c2ccc(C(=O)c4ccccc4)cc2)CO3)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 6/20 0.51
SCN9A Q15858 6/20 0.51
SCN5A Q14524 5/20 0.51
DRD2 P14416 3/20 0.42
DRD3 P35462 3/20 0.42
HTR2A P28223 2/20 0.42
ALDH1A1 P00352 2/20 0.39
GAA P10253 2/20 0.39
LMNA P02545 1/20 0.39
POLB P06746 1/20 0.39
MAPK1 P28482 1/20 0.39
EZH2 Q15910 1/20 0.39
KDM4E B2RXH2 1/20 0.38
HSD17B10 Q99714 1/20 0.38
HSP90AA1 P07900 1/20 0.38
HSP90AB1 P08238 1/20 0.38
WDR5 P61964 1/20 0.38
JAK3 P52333 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6932612 1.00 KCNH2 (0.51) KCNH2SCN9ASCN5ADRD2DRD3
SCHEMBL8064360 0.80 ALDH1A1 (0.38) ALDH1A1GAALMNAKDM4EHSD17B10
SCHEMBL6926134 0.78 KCNH2 (0.54) KCNH2SCN9ASCN5AALDH1A1LMNA
SCHEMBL6926137 0.78 KCNH2 (0.54) KCNH2SCN9ASCN5AALDH1A1LMNA
SCHEMBL6930424 0.76 ALDH1A1 (0.43) DRD2DRD3HTR2AALDH1A1LMNA
SCHEMBL6930432 0.76 ALDH1A1 (0.43) DRD2DRD3HTR2AALDH1A1LMNA
SCHEMBL8072714 0.75 KCNH2 (0.49) KCNH2SCN9ASCN5ADRD2ALDH1A1
SCHEMBL6820090 0.75 KCNH2 (0.51) KCNH2SCN9ASCN5AHTR2AWDR5
SCHEMBL6820074 0.75 KCNH2 (0.51) KCNH2SCN9ASCN5AHTR2AWDR5
SCHEMBL7022204 0.74 MTNR1A (0.60) KCNH2SCN9ASCN5ADRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1025096-B1 SUBSTITUTED CHROMAN DERIVATIVES ASTRAZENECA AB (SE) 2003-11-26 EP disclosed
US-6387899-B1 ANTISEROTONINE AGENTS; ANTIDEPRESSANTS ASTRAZENECA AB (SE) 2002-05-14 US disclosed
US-6384225-B1 5-PIPERIDINYL- OR PIPERAZINYL-SUBSTITUTED 3,4-DIHYDRO-2H-1-BENZOPYRANS ASTRAZENECA AB (SE) 2002-05-07 US disclosed