SCHEMBL6933869

SCHEMBL6933869

COc1ccc(C=C(C)N2CCNCC2)c(OC)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.50
KDM4E B2RXH2 1/20 0.50
LMNA P02545 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
CYP1A2 P05177 7/20 0.47
CYP1A1 P04798 6/20 0.47
CYP1B1 Q16678 6/20 0.47
ALDH1A1 P00352 4/20 0.45
KMT2A Q03164 3/20 0.44
MEN1 O00255 2/20 0.43
MAPT P10636 1/20 0.43
NFE2L2 Q16236 2/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
HTR3A P46098 2/20 0.43
HTR3E A5X5Y0 1/20 0.43
HTR3B O95264 1/20 0.43
HTR3D Q70Z44 1/20 0.43
HTR3C Q8WXA8 1/20 0.43
NCF1 P14598 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6931605 0.82 HTR3A (0.49) KDM4ELMNASMN1; SMN2ALDH1A1KMT2A
SCHEMBL4866793 0.76 KMT2A (0.44) CYP1A2CYP1A1CYP1B1ALDH1A1KMT2A
SCHEMBL6931871 0.75 TDP1 (0.50) GAAKDM4ESMN1; SMN2CYP1A2CYP1A1
SCHEMBL27567539 0.74 CYP1A2 (0.66) KDM4ECYP1A2CYP1A1CYP1B1ALDH1A1
SCHEMBL4753301 0.72 TSHR (0.59) KDM4ELMNAALDH1A1KMT2AMEN1
SCHEMBL6933867 0.70 ALDH1A1 (0.47) GAAKDM4ESMN1; SMN2ALDH1A1KMT2A
SCHEMBL27909079 0.70 JUN (0.44) GAAKDM4ELMNASMN1; SMN2CYP1A2
SCHEMBL7192327 0.70 CYP1A2 (0.63) GAAKDM4ECYP1A2CYP1A1CYP1B1
SCHEMBL6909563 0.69 ALDH1A1 (0.64) GAAKDM4ESMN1; SMN2CYP1A2CYP1A1
SCHEMBL233151 0.69 HTR3A (0.71) LMNAKMT2AMAPTHTR3AHTR3E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1366030-A2 MELANIN CONCENTRATING HORMONE RECEPTOR LIGANDS Neurogen Corporation (US) 2003-12-03 EP claimed
WO-2002004433-A2 MELANIN CONCENTRATING HORMONE RECEPTOR LIGANDS NEUROGEN CORPORATION (US) 2002-01-17 WO claimed