SCHEMBL6931871

SCHEMBL6931871

COc1ccc(C=C(C)N2CCNCC2)cc1OC

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.50
GAA P10253 1/20 0.50
ALDH1A1 P00352 3/20 0.49
KDM4E B2RXH2 2/20 0.49
KMT2A Q03164 2/20 0.49
L3MBTL1 Q9Y468 1/20 0.47
PTGS1 P23219 2/20 0.47
PTGS2 P35354 2/20 0.47
NQO2 P16083 1/20 0.47
HPGD P15428 1/20 0.43
ALOX15 P16050 1/20 0.43
MAPK1 P28482 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HSD17B10 Q99714 1/20 0.43
TSHR P16473 1/20 0.42
NFE2L2 Q16236 1/20 0.42
CYP1A1 P04798 1/20 0.42
CYP1A2 P05177 1/20 0.42
MEN1 O00255 1/20 0.41
ABCG2 Q9UNQ0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27926949 0.80 TDP1 (0.50) TDP1GAAALDH1A1KDM4EKMT2A
SCHEMBL11469832 0.78 KDM4E (0.80) TDP1ALDH1A1KDM4EKMT2AL3MBTL1
SCHEMBL11469833 0.78 KDM4E (0.80) TDP1ALDH1A1KDM4EKMT2AL3MBTL1
SCHEMBL6931605 0.75 HTR3A (0.49) ALDH1A1KDM4EKMT2AHPGDSMN1; SMN2
SCHEMBL29253491 0.75 ADRB1 (0.46) ALDH1A1KDM4EKMT2AHPGDSMN1; SMN2
SCHEMBL6933869 0.75 GAA (0.50) GAAALDH1A1KDM4EKMT2ASMN1; SMN2
SCHEMBL4871242 0.75 PTGS1 (0.42) TDP1GAAALDH1A1KDM4EKMT2A
SCHEMBL6933020 0.74 ADRB1 (0.47) TDP1L3MBTL1PTGS1PTGS2SMN1; SMN2
SCHEMBL6932180 0.73 SIGMAR1 (0.47) ALDH1A1KMT2AHPGDALOX15SMN1; SMN2
SCHEMBL6934619 0.72 CYP1A2 (0.46) TDP1ALDH1A1KDM4EKMT2APTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1366030-A2 MELANIN CONCENTRATING HORMONE RECEPTOR LIGANDS Neurogen Corporation (US) 2003-12-03 EP claimed
WO-2002004433-A2 MELANIN CONCENTRATING HORMONE RECEPTOR LIGANDS NEUROGEN CORPORATION (US) 2002-01-17 WO claimed