SCHEMBL6934203

SCHEMBL6934203

CN(C)CC1=C(c2cccc(O)c2)CC(c2ccccc2)CCC1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 1/20 0.39
HTR7 P34969 1/20 0.36
SIGMAR1 Q99720 3/20 0.36
DRD4 P21917 2/20 0.36
DRD3 P35462 2/20 0.36
DRD2 P14416 2/20 0.36
NFKB1 P19838 1/20 0.36
PRCP P42785 1/20 0.36
EBP Q15125 1/20 0.36
HRH3 Q9Y5N1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7870761 0.99 OPRK1 (0.39) OPRK1HTR7SIGMAR1DRD4DRD3
SCHEMBL6934590 0.94 DRD3 (0.41) SIGMAR1DRD4DRD3DRD2NFKB1
SCHEMBL6937110 0.93 ESR2 (0.37) OPRK1SIGMAR1DRD4DRD3DRD2
Hydrochloric Acid SCHEMBL7874356 0.93 DRD3 (0.40) SIGMAR1DRD4DRD3DRD2NFKB1
Hydrochloric Acid SCHEMBL7872662 0.92 ESR2 (0.36) OPRK1SIGMAR1DRD4DRD3DRD2
SCHEMBL6936489 0.90 PRKCZ (0.39) OPRK1SIGMAR1DRD4DRD3DRD2
SCHEMBL6937298 0.90 MAP1LC3B (0.39) SIGMAR1DRD4DRD3DRD2NFKB1
Hydrochloric Acid SCHEMBL7865265 0.89 MAP1LC3B (0.38) SIGMAR1DRD4DRD3DRD2NFKB1
Hydrochloric Acid SCHEMBL7870791 0.89 PRKCZ (0.38) OPRK1SIGMAR1DRD4DRD3DRD2
SCHEMBL6935012 0.88 HSD17B1 (0.39) OPRK1SIGMAR1DRD4DRD3DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1010689-B1 Substituted cycloheptenes, their preparation and use GRUENENTHAL GMBH (DE) 2003-01-15 EP claimed
EP-1010689-A1 Substituted cycloheptenes, their preparation and use Grünenthal GmbH (DE) 2000-06-21 EP claimed
EP-1010689-B1 Substituted cycloheptenes, their preparation and use GRUENENTHAL GMBH (DE) 2003-01-15 EP disclosed
EP-1010689-A1 Substituted cycloheptenes, their preparation and use Grünenthal GmbH (DE) 2000-06-21 EP disclosed