SCHEMBL6935012

SCHEMBL6935012

CN(C)CC1=C(c2cccc(O)c2)CC(c2ccc3ccccc3c2)CCC1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 1/20 0.39
HSD17B2 P37059 1/20 0.39
SLC6A4 P31645 8/20 0.38
SLC6A3 Q01959 7/20 0.38
SLC6A2 P23975 5/20 0.38
HRH3 Q9Y5N1 2/20 0.37
LSS P48449 1/20 0.35
DRD2 P14416 2/20 0.34
OPRK1 P41145 1/20 0.33
PFKFB3 Q16875 1/20 0.33
SIGMAR1 Q99720 3/20 0.33
DRD4 P21917 2/20 0.33
DRD3 P35462 2/20 0.33
NFKB1 P19838 1/20 0.33
PRCP P42785 1/20 0.33
EBP Q15125 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7874328 0.99 HSD17B1 (0.38) HSD17B1HSD17B2SLC6A4SLC6A3SLC6A2
SCHEMBL6940430 0.95 SLC6A2 (0.42) HSD17B1HSD17B2SLC6A4SLC6A3SLC6A2
SCHEMBL6934590 0.89 DRD3 (0.41) DRD2SIGMAR1DRD4DRD3NFKB1
SCHEMBL6934203 0.88 OPRK1 (0.39) HRH3DRD2OPRK1SIGMAR1DRD4
Hydrochloric Acid SCHEMBL7874356 0.88 DRD3 (0.40) DRD2SIGMAR1DRD4DRD3NFKB1
SCHEMBL6937110 0.88 ESR2 (0.37) HSD17B1HSD17B2HRH3DRD2OPRK1
Hydrochloric Acid SCHEMBL7872662 0.87 ESR2 (0.36) HSD17B1HSD17B2HRH3DRD2OPRK1
Hydrochloric Acid SCHEMBL7870761 0.87 OPRK1 (0.39) HRH3DRD2OPRK1SIGMAR1DRD4
SCHEMBL6936489 0.85 PRKCZ (0.39) HSD17B1HSD17B2HRH3LSSDRD2
SCHEMBL6937298 0.85 MAP1LC3B (0.39) DRD2SIGMAR1DRD4DRD3NFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1010689-B1 Substituted cycloheptenes, their preparation and use GRUENENTHAL GMBH (DE) 2003-01-15 EP claimed
EP-1010689-A1 Substituted cycloheptenes, their preparation and use Grünenthal GmbH (DE) 2000-06-21 EP claimed
EP-1010689-B1 Substituted cycloheptenes, their preparation and use GRUENENTHAL GMBH (DE) 2003-01-15 EP disclosed
EP-1010689-A1 Substituted cycloheptenes, their preparation and use Grünenthal GmbH (DE) 2000-06-21 EP disclosed