SCHEMBL6935178

SCHEMBL6935178

CCCCOc1ccc2c(c1)C(NS(C)(=O)=O)CC2(C)C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
KCNE1 P15382 2/20 0.42
KCNQ1 P51787 2/20 0.42
MMP1 P03956 6/20 0.39
MMP3 P08254 4/20 0.39
MMP13 P45452 4/20 0.39
MMP7 P09237 2/20 0.39
MMP2 P08253 2/20 0.39
MMP9 P14780 2/20 0.38
ADAM17 P78536 2/20 0.37
TSHR P16473 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
MAPK1 P28482 1/20 0.36
RECQL P46063 1/20 0.36
CRBN Q96SW2 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA7 P43166 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7464900 0.81 KCNE1 (0.52) NPC1RAB9AKCNE1KCNQ1MMP1
SCHEMBL6936617 0.78 KCNE1 (0.53) NPC1RAB9AKCNE1KCNQ1MMP1
SCHEMBL6932420 0.77 KCNE1 (0.45) NPC1RAB9AKCNE1KCNQ1MMP1
SCHEMBL6936603 0.76 LTA4H (0.38) NPC1RAB9AKCNE1KCNQ1TSHR
SCHEMBL26028475 0.65 KCNE1 (0.42) NPC1RAB9AKCNE1KCNQ1TSHR
SCHEMBL26029578 0.65 HRH3 (0.58) NPC1RAB9ATSHRL3MBTL1MAPK1
SCHEMBL14113144 0.64 NPC1 (0.93) NPC1RAB9ATSHRMAPK1RECQL
SCHEMBL6938514 0.64 ALDH1A1 (0.47) NPC1RAB9AL3MBTL1CA12CA1
SCHEMBL10071518 0.62 HRH3 (0.55) NPC1RAB9ATSHRL3MBTL1CA12
SCHEMBL5860140 0.61 PPARG (0.56) TSHRCA12CA1CA2CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0915087-B1 Sulfonamide substituted fused five-membered ring compounds, their use as medicaments as well as pharmaceutical compositions containing them AVENTIS PHARMA GMBH (DE) 2003-04-02 EP disclosed
US-6015822-A ANTIULCER, ANTIDIARRHEA, AND ANTIARRHYTHMIA AGENTS; CARDIOVASCULAR AND GASTROINTESTINAL DISORDERS HOECHST MARION ROUSSEL DEUTSCHLAND GMBH (DE) 2000-01-18 US disclosed
EP-0915087-A2 Sulfonamide substituted fused five-membered ring compounds, their use as medicaments as well as pharmaceutical compositions containing them Hoechst Marion Roussel Deutschland GmbH (DE) 1999-05-12 EP disclosed