SCHEMBL6935322

SCHEMBL6935322

CCCCN(C1CS(=O)(=O)c2cc([N+](=O)[O-])ccc21)S(C)(=O)=O

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 7/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
MAPT P10636 2/20 0.38
HTT P42858 4/20 0.35
ALDH1A1 P00352 3/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
NPSR1 Q6W5P4 1/20 0.35
LMNA P02545 1/20 0.35
VCAM1 P19320 1/20 0.33
SLC10A2 Q12908 1/20 0.33
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6937812 0.79 SLC10A2 (0.37) CA1CA2CA9MAPTSLC10A2
SCHEMBL6936648 0.75 CYP19A1 (0.40) CYP19A1MAPTHTTALDH1A1SMN1; SMN2
SCHEMBL6342196 0.72 CYP19A1 (0.37) CYP19A1MAPT
SCHEMBL8180505 0.71 CYP19A1 (0.42) CYP19A1MAPTALDH1A1KDM4E
SCHEMBL7132538 0.65 GAA (0.42) CYP19A1CA1CA2CA9HTT
SCHEMBL7434488 0.64 CYP1A2 (0.40) CA9MAPTHTTALDH1A1
SCHEMBL7434324 0.63 ALDH1A1 (0.38) CA1CA2CA9MAPTHTT
SCHEMBL14228900 0.60 CA12 (0.62) CA1CA2CA9MAPTHTT
SCHEMBL11117458 0.60 LMNA (0.58) CA1CA9MAPTHTTALDH1A1
Dinitrophenylene SCHEMBL27897921 0.59 TSHR (0.71) MAPTHTTALDH1A1SMN1; SMN2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0915087-B1 Sulfonamide substituted fused five-membered ring compounds, their use as medicaments as well as pharmaceutical compositions containing them AVENTIS PHARMA GMBH (DE) 2003-04-02 EP disclosed
US-6015822-A ANTIULCER, ANTIDIARRHEA, AND ANTIARRHYTHMIA AGENTS; CARDIOVASCULAR AND GASTROINTESTINAL DISORDERS HOECHST MARION ROUSSEL DEUTSCHLAND GMBH (DE) 2000-01-18 US disclosed
EP-0915087-A2 Sulfonamide substituted fused five-membered ring compounds, their use as medicaments as well as pharmaceutical compositions containing them Hoechst Marion Roussel Deutschland GmbH (DE) 1999-05-12 EP disclosed