SCHEMBL6937424

SCHEMBL6937424

CN(C)c1ccccc1CC1CCCCC1(O)Cc1ccc(F)cc1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 10/20 0.44
AQP1 P29972 1/20 0.33
SLC6A9 P48067 1/20 0.32
SLC6A2 P23975 3/20 0.32
SLC6A4 P31645 3/20 0.32
OPRM1 P35372 2/20 0.32
MEN1 O00255 1/20 0.32
OPRD1 P41143 1/20 0.32
OPRK1 P41145 1/20 0.32
KMT2A Q03164 1/20 0.32
ESR1 P03372 1/20 0.32
PGR P06401 1/20 0.32
HTR2A P28223 1/20 0.32
SLC6A3 Q01959 1/20 0.32
TRPC5 Q9UL62 1/20 0.32
CACNA1G O43497 1/20 0.32
TMEM97 Q5BJF2 2/20 0.31
SIGMAR1 Q99720 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6936768 0.91 SLC6A9 (0.39) TRPA1SLC6A9SLC6A2SLC6A4OPRM1
Hydrochloric Acid SCHEMBL7741185 0.90 OPRL1 (0.39) TRPA1SLC6A9SLC6A2SLC6A4OPRM1
SCHEMBL5846320 0.89 SLC6A4 (0.36) TRPA1SLC6A9SLC6A2SLC6A4OPRM1
SCHEMBL5845144 0.88 TRPA1 (0.35) TRPA1SLC6A2SLC6A4OPRM1MEN1
SCHEMBL6937427 0.88 TRPA1 (0.38) TRPA1SLC6A2SLC6A4OPRM1MEN1
Hydrochloric Acid SCHEMBL5847568 0.88 SLC6A4 (0.36) TRPA1SLC6A9SLC6A2SLC6A4OPRM1
Hydrochloric Acid SCHEMBL5846909 0.87 TRPA1 (0.34) TRPA1SLC6A2SLC6A4OPRM1MEN1
SCHEMBL6939736 0.87 SLC6A4 (0.40) SLC6A2SLC6A4OPRM1MEN1OPRD1
SCHEMBL6937028 0.86 TRPA1 (0.38) TRPA1SLC6A2SLC6A4OPRM1MEN1
SCHEMBL6939845 0.86 TRPA1 (0.38) TRPA1SLC6A2SLC6A4OPRM1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1043307-B1 3-amino-3-arylpropan-1-ol-derivates, their preparation and their use GRUENENTHAL GMBH (DE) 2003-06-04 EP claimed
US-6410790-B1 ANALGESICS GRUENENTHAL GMBH (DE) 2002-06-25 US claimed
US-6410790-B1 ANALGESICS GRUENENTHAL GMBH (DE) 2002-06-25 US disclosed